SCHEMBL8083649

SCHEMBL8083649

CCOP(=O)(CNc1cc(OCc2ccccc2)c(C(F)(F)F)cc1N)OCC

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
S1PR1 P21453 2/20 0.37
S1PR4 O95977 1/20 0.37
S1PR3 Q99500 1/20 0.37
S1PR5 Q9H228 1/20 0.37
MRGPRX4 Q96LA9 4/20 0.36
RXRA P19793 2/20 0.36
RXRB P28702 2/20 0.36
RXRG P48443 2/20 0.36
HDAC1 Q13547 2/20 0.35
HDAC3 O15379 1/20 0.35
HDAC2 Q92769 1/20 0.35
HDAC8 Q9BY41 1/20 0.35
MEN1 O00255 1/20 0.34
MAPT P10636 1/20 0.34
KMT2A Q03164 1/20 0.34
BRD4 O60885 3/20 0.34
ALOX5AP P20292 1/20 0.34
HTR1A P08908 1/20 0.33
ADRA1D P25100 1/20 0.33
ADRA1A P35348 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8098268 0.85 SMN1; SMN2 (0.35) HDAC1HDAC3HDAC2HDAC8MAPT
SCHEMBL8090679 0.85 MAPT (0.43) MEN1MAPTKMT2AHTR1AADRA1D
SCHEMBL8083652 0.81 PPARG (0.36) S1PR1S1PR4S1PR3S1PR5MRGPRX4
SCHEMBL8098486 0.80 AR (0.35) S1PR1HDAC1HDAC3HDAC2HDAC8
SCHEMBL8098731 0.80 CYP1A2 (0.34) MEN1KMT2A
SCHEMBL8083938 0.79 RHOC (0.35) HDAC1MEN1MAPTKMT2A
SCHEMBL8604509 0.78 L3MBTL1 (0.41) MAPT
SCHEMBL8098784 0.78 NPSR1 (0.39) MEN1MAPTKMT2A
SCHEMBL8602899 0.76 ALDH1A1 (0.39) S1PR1S1PR4S1PR3S1PR5HDAC1
SCHEMBL8090772 0.74 PTGER4 (0.41) HDAC1MEN1MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136805-A Quinoxaline dione derivatives, their production and their use in medicaments SCNERING AKTIENGESELLSCHAFT (DE) 2000-10-24 US disclosed