SCHEMBL8083709

SCHEMBL8083709

O=P(O)(Cc1ccncc1)Oc1ccccc1

nearest known ligand 0.55

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP19A1 P11511 1/20 0.49
SRC P12931 1/20 0.48
HTT P42858 3/20 0.45
SMN1; SMN2 Q16637 3/20 0.45
ALPL P05186 1/20 0.45
ALPI P09923 1/20 0.45
ALPG P10696 1/20 0.45
LMNA P02545 2/20 0.44
CYP3A4 P08684 1/20 0.44
MMP13 P45452 1/20 0.44
MAPK14 Q16539 1/20 0.44
ANPEP P15144 2/20 0.43
LAP3 P28838 2/20 0.43
KLK8 O60259 1/20 0.42
PLAU P00749 1/20 0.42
KLK2 P20151 1/20 0.42
KLK4 Q9Y5K2 1/20 0.42
FDPS P14324 1/20 0.41
CYP2C9 P11712 1/20 0.41
CYP2C19 P33261 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3836998 0.88 SRC (0.57) SRCHTTANPEPLAP3KLK8
SCHEMBL916423 0.80 SRC (0.48) SRCHTTLMNAANPEPLAP3
SCHEMBL27882402 0.79 LMNA (0.52) SRCHTTLMNAANPEPLAP3
SCHEMBL8046728 0.77 CXCL8 (0.46) CYP19A1HTTSMN1; SMN2ALPLALPI
SCHEMBL27882400 0.77 MAOA (0.47) SRCSMN1; SMN2ANPEPLAP3KLK8
SCHEMBL22321983 0.77 SRC (0.44) SRCHTTLMNAANPEPLAP3
SCHEMBL22321985 0.77 ALDH1A1 (0.50) SRCHTTSMN1; SMN2PLAU
SCHEMBL13538164 0.75 CA1 (0.55) SRCHTTSMN1; SMN2LMNACYP3A4
SCHEMBL16238910 0.74 ALDH1A1 (0.49) SRCHTTSMN1; SMN2L3MBTL1
SCHEMBL27882575 0.73 PARP10 (0.56) CYP3A4ANPEPLAP3KLK8PLAU

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1044206-A1 PRODRUGS OF NAALADASE INHIBITORS Guildford Pharmaceuticals Inc. (US) 2000-10-18 EP disclosed
WO-1999033849-A1 PRODRUGS OF NAALADASE INHIBITORS GUILDFORD PHARMACEUTICALS INC. (US) 1999-07-08 WO disclosed