SCHEMBL8083716

SCHEMBL8083716

CCC(C)OP(=O)(O)CNc1cc(-c2ccc(OC)cc2)c(C(F)(F)F)cc1N

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
AKR1C3 P42330 3/20 0.37
AKR1C2 P52895 3/20 0.37
AKR1C4 P17516 2/20 0.35
AKR1C1 Q04828 2/20 0.35
AKR1B10 O60218 1/20 0.35
DHODH Q02127 1/20 0.34
TP53 P04637 3/20 0.33
EPHX2 P34913 2/20 0.33
CFTR P13569 1/20 0.33
FFAR4 Q5NUL3 1/20 0.33
PTGDR2 Q9Y5Y4 1/20 0.32
WDR5 P61964 1/20 0.32
MEN1 O00255 2/20 0.32
KMT2A Q03164 2/20 0.32
ABCG2 Q9UNQ0 1/20 0.32
SRD5A2 P31213 1/20 0.32
NPC1 O15118 2/20 0.32
RAB9A P51151 2/20 0.32
HSD17B10 Q99714 2/20 0.32
MAPK1 P28482 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8181084 0.84 CFTR (0.51) CFTRWDR5SMN1; SMN2KDM4EALDH1A1
SCHEMBL8083711 0.81 FFAR4 (0.36) AKR1C3AKR1C2AKR1C4AKR1C1AKR1B10
SCHEMBL8098272 0.79 UBE2M (0.34) DHODHEPHX2HPGDPPARG
SCHEMBL8083940 0.77 RHOC (0.36) MEN1KMT2ANPC1KDM4EALDH1A1
SCHEMBL8098790 0.76 NPSR1 (0.36) DHODHKDM4EALDH1A1MAPT
SCHEMBL8090776 0.76 PTGER4 (0.38) EPHX2MEN1KMT2AMAPK1SMN1; SMN2
SCHEMBL8083652 0.75 PPARG (0.36) MEN1KMT2AMAPTPPARG
SCHEMBL8342163 0.75 SERPINE1 (0.37) TP53NPC1RAB9ASMN1; SMN2KDM4E
SCHEMBL8345101 0.74 ALDH1A1 (0.41) TP53SMN1; SMN2KDM4EALDH1A1MAPT
SCHEMBL8098738 0.73 CYP1A2 (0.33)

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6136805-A Quinoxaline dione derivatives, their production and their use in medicaments SCNERING AKTIENGESELLSCHAFT (DE) 2000-10-24 US disclosed