SCHEMBL8084534

SCHEMBL8084534

CCC(COc1ccccc1)Nc1nc(Cl)nc(C(F)(F)F)n1

nearest known ligand 0.50

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.50
KDM4E B2RXH2 1/20 0.35
NFKB1 P19838 1/20 0.35
IDH1 O75874 1/20 0.34
IDH2 P48735 1/20 0.34
KCNH3 Q9ULD8 1/20 0.34
TLR7 Q9NYK1 1/20 0.34
GAA P10253 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
HTR7 P34969 1/20 0.33
MAOA P21397 1/20 0.33
PTGS1 P23219 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8070478 0.86 TSHR (0.43) ALDH1A1KDM4EHTR7MAOAPTGS1
SCHEMBL7613516 0.80 ALDH1A1 (0.38) ALDH1A1KCNH3
SCHEMBL11255273 0.72 APP (0.46) ALDH1A1KDM4ETLR7
SCHEMBL7676182 0.72 HTR2C (0.35) ALDH1A1KDM4EIDH1IDH2TDP1
SCHEMBL7960038 0.71 SCN9A (0.41) ALDH1A1TLR7
SCHEMBL6982625 0.70 TSHR (0.41) KDM4EGAAHTR7
SCHEMBL7946808 0.70 HTR7 (0.45) ALDH1A1KCNH3HTR7MAOAPTGS1
SCHEMBL8084532 0.66 ALDH1A1 (0.39) ALDH1A1TLR7TDP1
SCHEMBL11445845 0.65 MAOA (0.62) MAOAPTGS1
SCHEMBL7615960 0.64 CDK1 (0.32) ALDH1A1IDH1IDH2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1034168-A1 SUBSTITUTED ARYLOXY ALKYL AMINO TRIAZINES Bayer Aktiengesellschaft (DE) 2000-09-13 EP disclosed
WO-1999021841-A1 SUBSTITUTED ARYLOXY ALKYL AMINO TRIAZINES BAYER AKTIENGESELLSCHAFT (DE) 1999-05-06 WO disclosed