SCHEMBL8084539

SCHEMBL8084539

CC(=O)c1ccc2c(c1)C(n1nc(O)ccc1=O)=C(C)C(C)(C)O2

nearest known ligand 0.32

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
S100A4 P26447 1/20 0.32
KDM4E B2RXH2 2/20 0.31
ALDH1A1 P00352 2/20 0.31
SMN1; SMN2 Q16637 1/20 0.31
HSD17B1 P14061 1/20 0.30
POLB P06746 1/20 0.30
HPGD P15428 1/20 0.30
MAPT P10636 1/20 0.30
RECQL P46063 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090068 0.90 ALDH1A1 (0.34) KDM4EALDH1A1SMN1; SMN2POLBHPGD
SCHEMBL8088362 0.87 SLC9A1 (0.30)
SCHEMBL8085332 0.86 ALDH1A1 (0.46) ALDH1A1MAPTRECQL
SCHEMBL8084221 0.82
SCHEMBL8090648 0.81 ABCC9 (0.35) KDM4E
SCHEMBL8085297 0.81 MAPT (0.35) S100A4ALDH1A1POLBMAPT
SCHEMBL8077225 0.78 HSD17B1 (0.35) S100A4KDM4EALDH1A1SMN1; SMN2HSD17B1
SCHEMBL8088434 0.76 S100A4 (0.37) S100A4KDM4EALDH1A1SMN1; SMN2POLB
SCHEMBL9372349 0.69 RAB9A (0.37) ALDH1A1SMN1; SMN2POLBMAPT
SCHEMBL10697118 0.69 RAB9A (0.37) ALDH1A1SMN1; SMN2POLBMAPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed
EP-0340718-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1989-11-08 EP disclosed