SCHEMBL8084592

SCHEMBL8084592

COC(=O)Oc1cc(N)c(F)cc1Cl

nearest known ligand 0.46

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CUL4A Q13619 1/20 0.46
GAA P10253 3/20 0.43
NPC1 O15118 4/20 0.41
RAB9A P51151 3/20 0.39
MAPT P10636 3/20 0.39
KDM4E B2RXH2 4/20 0.37
POLB P06746 2/20 0.36
HPGD P15428 2/20 0.36
HSD17B10 Q99714 1/20 0.36
LMNA P02545 2/20 0.35
TP53 P04637 1/20 0.35
NPSR1 Q6W5P4 1/20 0.35
SMN1; SMN2 Q16637 5/20 0.35
ALDH1A1 P00352 3/20 0.35
KMT2A Q03164 2/20 0.35
ABL1 P00519 1/20 0.35
MEN1 O00255 1/20 0.35
GLA P06280 1/20 0.35
APEX1 P27695 1/20 0.34
RORC P51449 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8370837 0.90 NPC1 (0.37) CUL4AGAANPC1RAB9AMAPT
SCHEMBL8602332 0.86 RORC (0.35) CUL4AGAANPC1RAB9AMAPT
SCHEMBL7211056 0.85 KDM4E (0.40) CUL4AGAARAB9AMAPTKDM4E
SCHEMBL17466053 0.83 KDM4E (0.42) GAANPC1RAB9AMAPTKDM4E
SCHEMBL8600593 0.83 ELANE (0.36) CUL4AGAANPC1RAB9AMAPT
SCHEMBL8604258 0.83 CUL4A (0.49) CUL4AGAANPC1RAB9AMAPT
SCHEMBL8076435 0.83 TSHR (0.44) CUL4AMAPTHPGDLMNATP53
SCHEMBL6430813 0.82 KDM4E (0.38) CUL4AGAAMAPTKDM4EHPGD
SCHEMBL7219984 0.82 GAA (0.39) CUL4AGAANPC1RAB9AMAPT
SCHEMBL8602520 0.82 CUL4A (0.33) CUL4AGAANPC1MAPTHPGD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 15 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
JP-8169865-A None JP disclosed
EP-0493606-B1 HETEROCYCLE-SUBSTITUTED BENZENE DERIVATIVE, PRODUCTION THEREOF, AND HERBICIDE CONTAINING THE SAME AS ACTIVE INGREDIENT SAGAMI CHEM RES (JP) 2000-10-18 EP disclosed
EP-1006105-A1 Benzene derivatives SAGAMI CHEMICAL RESEARCH CENTER (JP) 2000-06-07 EP disclosed
EP-0626370-B1 Process for producing aromatic isothiocyanate derivatives SUMITOMO CHEMICAL CO (JP) 1998-02-11 EP disclosed
JP-H08169865-A DIHALOPHENYL CARBONATE DERIVATIVE SAGAMI CHEM RES CENTER 1996-07-02 JP disclosed
US-5464811-A Benzene derivatives substituted with heterocyclic ring and herbicides containing same as active ingredients SAGAMI CHEMICAL RESEARCH CENTER (JP) 1995-11-07 US disclosed
US-5424277-A An N-substituted-3,4,5,6-tetrahydrophthalimide derivative characterized by having a cycloalkoxy group at the 5-position of the phenyl ring on the nitrogen SAGAMI CHEMICAL RESEARCH CENTER (JP) 1995-06-13 US disclosed
EP-0626370-A1 Process for producing aromatic isothiocyanate derivatives SUMITOMO CHEMICAL COMPANY LIMITED (JP) 1994-11-30 EP disclosed
EP-0493606-A1 HETEROCYCLE-SUBSTITUTED BENZENE DERIVATIVE, PRODUCTION THEREOF, AND HERBICIDE CONTAINING THE SAME AS ACTIVE INGREDIENT SAGAMI CHEMICAL RESEARCH CENTER (JP) 1992-07-08 EP disclosed
EP-0262428-B1 HYDANTOIN DERIVATIVES AND HERBICIDES CONTAINING THE DERIVATIVES AS AN ACTIVE INGREDIENT SAGAMI CHEMICAL RESEARCH CENTER (JP) 1991-08-14 EP disclosed
EP-0440319-A1 Process and intermediates for the preparation of annelated iminothiazoles SCHERING AKTIENGESELLSCHAFT (DE) 1991-08-07 EP disclosed
US-5017213-A Herbicides NIHON TOKUSHU NOYAKU SEIZO K. K. (JP) 1991-05-21 US disclosed
US-4902337-A Herbicidal hydantoin derivatives SAGAMI CHEMICAL RESEARCH (JP) 1990-02-20 US disclosed
EP-0351641-A1 1-Phenylpyrrole NIHON BAYER AGROCHEM K.K. (JP) 1990-01-24 EP disclosed
EP-0262428-A1 Hydantoin derivatives and herbicides containing the derivatives as an active ingredient SAGAMI CHEMICAL RESEARCH CENTER (JP) 1988-04-06 EP disclosed