SCHEMBL8085303

SCHEMBL8085303

CC1(C)C=C(n2cc(Br)cc(Br)c2=O)c2cc([N+](=O)[O-])ccc2O1

nearest known ligand 0.34

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CHRM2 P08172 1/20 0.34
HTR1A P08908 1/20 0.34
ADRA2A P08913 1/20 0.34
DRD1 P21728 1/20 0.34
PTGS1 P23219 1/20 0.34
SLC6A4 P31645 1/20 0.34
DRD3 P35462 1/20 0.34
ALDH1A1 P00352 1/20 0.34
CYP3A4 P08684 1/20 0.34
TDP1 Q9NUW8 1/20 0.34
CHEK1 O14757 1/20 0.34
PIM1 P11309 1/20 0.34
LIMK1 P53667 1/20 0.34
TYRO3 Q06418 1/20 0.34
MAPK14 Q16539 1/20 0.34
CLK4 Q9HAZ1 1/20 0.34
PTPRC P08575 3/20 0.33
CASP3 P42574 2/20 0.33
S100A4 P26447 2/20 0.33
CASP1 P29466 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8084409 0.92 ALDH1A1 (0.35) CHRM2HTR1AADRA2ADRD1PTGS1
SCHEMBL8085257 0.90 MEN1 (0.34) CHRM2HTR1AADRA2ADRD1PTGS1
SCHEMBL8090154 0.89 TDP1 (0.34) CHRM2HTR1AADRA2ADRD1PTGS1
SCHEMBL8085225 0.89 TDP1 (0.36) CHRM2HTR1AADRA2ADRD1PTGS1
SCHEMBL8090476 0.84 SMN1; SMN2 (0.38) ALDH1A1CYP3A4TDP1MEN1KMT2A
SCHEMBL8084934 0.84 CFTR (0.38) ALDH1A1TDP1KMT2A
SCHEMBL8085338 0.82 KMT2A (0.38) CHRM2HTR1AADRA2ADRD1PTGS1
SCHEMBL8085331 0.81 HSD17B10 (0.38) CHRM2HTR1AADRA2ADRD1PTGS1
SCHEMBL8085035 0.81 ALDH1A1 (0.38) CHRM2HTR1AADRA2ADRD1PTGS1
SCHEMBL8085433 0.81 PDE4A (0.40) MALT1ABCC9

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
EP-0273262-A2 Chroman derivatives MERCK PATENT GmbH (DE) 1988-07-06 EP disclosed