SCHEMBL8206417

SCHEMBL8206417

CCC1(CC)C=C(n2cc([N+](=O)[O-])cc([N+](=O)[O-])c2=O)c2cc([N+](=O)[O-])ccc2O1

nearest known ligand 0.35

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 4/20 0.35
KMT2A Q03164 4/20 0.35
CASP1 P29466 1/20 0.34
CASP3 P42574 1/20 0.34
CASP4 P49662 1/20 0.34
CASP7 P55210 1/20 0.34
CASP9 P55211 1/20 0.34
CASP6 P55212 1/20 0.34
ADORA2B P29275 1/20 0.33
CHRM2 P08172 1/20 0.33
HTR1A P08908 1/20 0.33
ADRA2A P08913 1/20 0.33
DRD1 P21728 1/20 0.33
PTGS1 P23219 1/20 0.33
SLC6A4 P31645 1/20 0.33
DRD3 P35462 1/20 0.33
ALDH1A1 P00352 3/20 0.33
TDP1 Q9NUW8 2/20 0.33
CYP3A4 P08684 1/20 0.33
CYP1A2 P05177 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085338 0.87 KMT2A (0.38) MEN1KMT2ACASP1CASP3CASP4
SCHEMBL8089644 0.78 MEN1 (0.34) MEN1KMT2ACASP1CASP3CASP4
SCHEMBL8085257 0.78 MEN1 (0.34) MEN1KMT2ACASP1CASP3CASP4
SCHEMBL8088704 0.76 ABCC9 (0.40) MEN1KMT2ATDP1MALT1MAPK1
SCHEMBL8084409 0.75 ALDH1A1 (0.35) MEN1KMT2ACASP1CASP3CASP4
SCHEMBL8076960 0.75 MEN1 (0.37) MEN1KMT2ACASP1CASP3CASP4
SCHEMBL8085331 0.75 HSD17B10 (0.38) MEN1KMT2ACASP1CASP3CASP4
SCHEMBL8090699 0.73 ALDH1A1 (0.37) MEN1KMT2ACASP1CASP3CASP4
SCHEMBL7291279 0.73 ADORA2B (0.31) MEN1KMT2AADORA2BALDH1A1
SCHEMBL8085035 0.72 ALDH1A1 (0.38) MEN1KMT2ACASP1CASP3CASP4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed