SCHEMBL8090111

SCHEMBL8090111

CC1=C(n2cc(C(=O)O)ccc2=O)c2cc(C#N)ccc2OC1(C)C

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
RARA P10276 1/20 0.36
RARB P10826 1/20 0.36
RARG P13631 1/20 0.36
ABCC9 O60706 7/20 0.35
ALK Q9UM73 1/20 0.35
ABCC8 Q09428 2/20 0.34
KCNJ11 Q14654 2/20 0.34
KCNJ8 Q15842 2/20 0.34
ALDH1A1 P00352 1/20 0.34
MAPT P10636 1/20 0.34
RECQL P46063 1/20 0.34
CYP1A2 P05177 1/20 0.34
CYP2D6 P10635 1/20 0.34
CYP2C9 P11712 1/20 0.34
CYP2C19 P33261 1/20 0.34
LMNA P02545 1/20 0.34
MALT1 Q9UDY8 1/20 0.33
KDM4C Q9H3R0 1/20 0.33
ABCB1 P08183 2/20 0.32
KDM4E B2RXH2 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085328 0.86 ABCC9 (0.36) ABCC9ABCC8KCNJ11KCNJ8MAPT
SCHEMBL8077233 0.84 ABCC9 (0.40) ABCC9MALT1ABCB1
SCHEMBL7267033 0.84 MALT1 (0.35) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL7276803 0.84 DRD2 (0.37) ABCC9ALDH1A1CYP2C19KDM4E
SCHEMBL8084525 0.82 ABCC9 (0.40) ABCC9MAPTMALT1ABCB1
SCHEMBL8090686 0.82 CA9 (0.42) ALDH1A1MALT1
SCHEMBL8077161 0.80 PDE4A (0.40) RARARARBRARGABCC9ALK
SCHEMBL7267575 0.80 ABCC9 (0.37) ABCC9ABCC8KCNJ11KCNJ8CYP1A2
SCHEMBL8085086 0.79 MALT1 (0.35) ABCC9ABCC8KCNJ11KCNJ8MAPT
SCHEMBL8077117 0.79 ABCC9 (0.36) RARARARBRARGABCC9ABCC8

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed
EP-0340718-A1 Chroman derivatives MERCK PATENT GmbH (DE) 1989-11-08 EP disclosed