SCHEMBL8077233

SCHEMBL8077233

CC1=C(n2cc(Cl)ccc2=O)c2cc(C#N)ccc2OC1(C)C

nearest known ligand 0.40

Predicted protein targets (top 5)

geneUniProtsupporting neighboursconfidence
ABCC9 O60706 13/20 0.40
MALT1 Q9UDY8 1/20 0.35
MIF P14174 2/20 0.34
ABCB1 P08183 2/20 0.32
CASP3 P42574 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8085328 0.87 ABCC9 (0.36) ABCC9MALT1ABCB1CASP3
SCHEMBL7267033 0.87 MALT1 (0.35) ABCC9MALT1ABCB1CASP3
SCHEMBL8076916 0.86 ABCC9 (0.38) ABCC9MALT1MIFABCB1
SCHEMBL7267575 0.84 ABCC9 (0.37) ABCC9MALT1ABCB1CASP3
SCHEMBL8085360 0.84 ABCC9 (0.37) ABCC9MALT1MIFABCB1
SCHEMBL8090111 0.84 RARA (0.36) ABCC9MALT1ABCB1
SCHEMBL8084525 0.84 ABCC9 (0.40) ABCC9MALT1ABCB1
SCHEMBL7276803 0.83 DRD2 (0.37) ABCC9
SCHEMBL8085086 0.81 MALT1 (0.35) ABCC9MALT1ABCB1CASP3
SCHEMBL8084273 0.81 VCAM1 (0.38) ABCC9MALT1MIF

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6153627-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-28 US disclosed
US-6040308-A Chroman derivatives MERCK GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-03-21 US disclosed
US-5387587-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1995-02-07 US disclosed
US-5013853-A Chroman derivatives MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 1991-05-07 US disclosed