SCHEMBL8090195

SCHEMBL8090195

CS(=O)(=O)C1(c2cc(N)nc(-c3ccc(NC(=O)Nc4ccon4)cc3)n2)CC1

nearest known ligand 0.47

Predicted protein targets (top 10)

geneUniProtsupporting neighboursconfidence
RAB9A P51151 3/20 0.47
POLB P06746 1/20 0.47
NPC1 O15118 1/20 0.44
MTOR P42345 2/20 0.44
KMT2A Q03164 3/20 0.43
MEN1 O00255 2/20 0.43
PIK3CD O00329 6/20 0.39
ATR Q13535 2/20 0.38
PIK3CA P42336 3/20 0.37
KDR P35968 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8099967 0.88 RAB9A (0.41) RAB9APOLBNPC1MTORKMT2A
SCHEMBL8095575 0.87 ALDH1A1 (0.49) RAB9ANPC1KMT2AMEN1PIK3CD
SCHEMBL8084988 0.87 RAB9A (0.41) RAB9APOLBNPC1MTORKMT2A
SCHEMBL8091838 0.86 KMT2A (0.43) RAB9APOLBNPC1MTORKMT2A
SCHEMBL8091635 0.85 ATR (0.47) RAB9ANPC1MTORKMT2AMEN1
SCHEMBL8093540 0.85 RAB9A (0.39) RAB9APOLBNPC1MTORKMT2A
SCHEMBL8097448 0.84 PIK3CA (0.43) MTORKMT2AMEN1PIK3CDATR
SCHEMBL8092389 0.84 PIK3CD (0.37) RAB9ANPC1MTORKMT2APIK3CD
SCHEMBL8083616 0.82 ATR (0.42) MTORKMT2AMEN1PIK3CDATR
SCHEMBL8098188 0.82 CA12 (0.44) MTORKMT2AMEN1PIK3CDATR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed