SCHEMBL8083973

SCHEMBL8083973

CNC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccc(F)cc4)CC3)n2)cc1

nearest known ligand 0.43

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.43
PIK3CA P42336 4/20 0.41
MTOR P42345 3/20 0.41
KMT2A Q03164 2/20 0.40
CA2 P00918 5/20 0.40
CA9 Q16790 5/20 0.40
CA12 O43570 4/20 0.40
CA1 P00915 4/20 0.40
CA4 P22748 1/20 0.40
CA7 P43166 1/20 0.40
PIK3CG P48736 2/20 0.39
TP53 P04637 1/20 0.39
NAMPT P43490 1/20 0.39
KDM1A O60341 1/20 0.37
MEN1 O00255 1/20 0.37
NPC1 O15118 1/20 0.37
RAB9A P51151 1/20 0.37
GAA P10253 1/20 0.36
PIP4K2A P48426 1/20 0.36
PIP4K2B P78356 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8089917 0.93 PIK3CA (0.39) ALDH1A1PIK3CAMTORKMT2ACA2
SCHEMBL8092637 0.92 KMT2A (0.42) PIK3CAMTORKMT2ACA2CA9
SCHEMBL8097257 0.91 ALDH1A1 (0.41) ALDH1A1PIK3CAMTORKMT2ACA2
SCHEMBL8097712 0.91 KMT2A (0.39) PIK3CAMTORKMT2ACA2CA9
SCHEMBL8090246 0.90 PIK3CA (0.42) ALDH1A1PIK3CAMTORKMT2APIK3CG
SCHEMBL8083334 0.90 CA1 (0.41) ALDH1A1PIK3CAMTORKMT2ACA2
SCHEMBL8099749 0.90 MTOR (0.40) PIK3CAMTORKMT2APIK3CGNAMPT
SCHEMBL8083200 0.89 ALDH1A1 (0.43) ALDH1A1PIK3CAMTORKMT2ACA2
SCHEMBL8094619 0.89 PIP4K2A (0.40) PIK3CAMTORKMT2APIK3CGNAMPT
SCHEMBL8094423 0.88 CA2 (0.43) ALDH1A1PIK3CAMTORKMT2ACA2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed