SCHEMBL8097257

SCHEMBL8097257

CNC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccc(C)cc4)CC3)n2)cc1

nearest known ligand 0.45

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 1/20 0.41
KMT2A Q03164 2/20 0.41
MEN1 O00255 1/20 0.41
LMNA P02545 1/20 0.41
HPGD P15428 1/20 0.41
PTPN7 P35236 1/20 0.40
RAB9A P51151 1/20 0.40
CA2 P00918 2/20 0.40
CA4 P22748 2/20 0.40
CA9 Q16790 2/20 0.40
PIK3CA P42336 2/20 0.39
MTOR P42345 2/20 0.39
PIK3CG P48736 2/20 0.39
CA12 O43570 1/20 0.39
CA1 P00915 1/20 0.39
CA6 P23280 1/20 0.39
CA5A P35218 1/20 0.39
CA7 P43166 1/20 0.39
CA13 Q8N1Q1 1/20 0.39
CA14 Q9ULX7 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8092637 0.93 KMT2A (0.42) KMT2ACA2CA9PIK3CAMTOR
SCHEMBL8083973 0.91 ALDH1A1 (0.43) ALDH1A1KMT2AMEN1RAB9ACA2
SCHEMBL8090246 0.91 PIK3CA (0.42) ALDH1A1KMT2AMEN1HPGDPIK3CA
SCHEMBL8099749 0.90 MTOR (0.40) KMT2APIK3CAMTORPIK3CG
SCHEMBL8097712 0.88 KMT2A (0.39) KMT2AMEN1CA2CA9PIK3CA
SCHEMBL8096342 0.88 PIK3CA (0.41) ALDH1A1KMT2AMEN1HPGDPIK3CA
SCHEMBL8089917 0.88 PIK3CA (0.39) ALDH1A1KMT2ACA2CA9PIK3CA
SCHEMBL8099632 0.87 CA1 (0.42) ALDH1A1KMT2AMEN1LMNAHPGD
SCHEMBL8093151 0.87 KMT2A (0.37) ALDH1A1KMT2AMEN1LMNARAB9A
SCHEMBL8097448 0.86 PIK3CA (0.43) ALDH1A1KMT2AMEN1HPGDPIK3CA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed