SCHEMBL8096681

SCHEMBL8096681

NC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccccn4)CC3)n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ATR Q13535 2/20 0.40
MTOR P42345 3/20 0.34
NAMPT P43490 3/20 0.34
MAOA P21397 1/20 0.34
MAPT P10636 4/20 0.33
MEN1 O00255 3/20 0.33
ALDH1A1 P00352 3/20 0.33
HPGD P15428 3/20 0.33
KMT2A Q03164 3/20 0.33
KDM4E B2RXH2 2/20 0.33
NPSR1 Q6W5P4 1/20 0.33
RXFP1 Q9HBX9 1/20 0.33
CYP2C19 P33261 1/20 0.33
IGF1R P08069 1/20 0.32
KDM1A O60341 1/20 0.32
MAOB P27338 1/20 0.32
ABCC9 O60706 1/20 0.32
ABCC8 Q09428 1/20 0.32
KCNJ11 Q14654 1/20 0.32
KCNJ8 Q15842 1/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8096070 0.90 MTOR (0.40) ATRMTORNAMPTMAOAKMT2A
SCHEMBL8092270 0.89 NPC1 (0.43) ATRMTORMAPTMEN1KMT2A
SCHEMBL8092294 0.87 ROCK2 (0.39) ATRMTORNAMPTIGF1RPIK3R1
SCHEMBL8098135 0.86 MTOR (0.39) ATRMTORNAMPTIGF1RAKT1
SCHEMBL8091293 0.86 MAPT (0.42) ATRMTORNAMPTMAPTMEN1
SCHEMBL8091129 0.86 KDR (0.40) ATRGAA
SCHEMBL8091924 0.86 NAMPT (0.39) ATRNAMPTPIK3CA
SCHEMBL8097714 0.85 NAMPT (0.39) ATRNAMPTMAPTKMT2AIGF1R
SCHEMBL8098769 0.85 NAMPT (0.39) ATRNAMPT
SCHEMBL8093540 0.84 RAB9A (0.39) ATRMTORMEN1KMT2AKDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed