SCHEMBL8091796

SCHEMBL8091796

CCS(=O)(=O)Cc1cc(N)nc(-c2ccc(NC(=O)Nc3ccccn3)cc2)n1

nearest known ligand 0.49

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
NPC1 O15118 7/20 0.49
RAB9A P51151 7/20 0.49
FLT3 P36888 2/20 0.46
SMN1; SMN2 Q16637 2/20 0.46
ADORA3 P0DMS8 1/20 0.46
PIM1 P11309 1/20 0.46
ADORA2A P29274 1/20 0.46
ADORA2B P29275 1/20 0.46
ADORA1 P30542 1/20 0.46
PIM3 Q86V86 1/20 0.46
AURKB Q96GD4 1/20 0.46
LIMK1 P53667 1/20 0.46
LMNA P02545 3/20 0.45
PIK3CA P42336 4/20 0.43
MTOR P42345 3/20 0.43
MEN1 O00255 1/20 0.43
KMT2A Q03164 1/20 0.43
KIT P10721 1/20 0.41
PDGFRA P16234 1/20 0.41
PIK3CD O00329 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8215437 0.84 PIK3CA (0.46) NPC1RAB9AFLT3SMN1; SMN2ADORA3
SCHEMBL8206190 0.81 PIK3CD (0.43) PIK3CAMTORMEN1KMT2APIK3CD
SCHEMBL8084637 0.81 CA12 (0.45) PIK3CAMTORMEN1KMT2APIK3CD
SCHEMBL8098332 0.81 PIK3CA (0.48) RAB9APIK3CAMTORMEN1KMT2A
SCHEMBL11925577 0.80 LMNA (0.45) NPC1RAB9AFLT3SMN1; SMN2ADORA3
SCHEMBL8205071 0.80 PIK3CA (0.54) LMNAPIK3CAMTORMEN1KMT2A
SCHEMBL8091882 0.79 PIK3CA (0.45) FLT3SMN1; SMN2AURKBLIMK1PIK3CA
SCHEMBL8217167 0.79 PIK3CA (0.40) PIK3CAMTORMEN1KMT2APIK3CD
SCHEMBL8217546 0.79 L3MBTL1 (0.55) NPC1RAB9ASMN1; SMN2PIK3CAMEN1
SCHEMBL13948517 0.79 PIK3CA (0.67) PIK3CAMTORPIK3CD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed