SCHEMBL8098751

SCHEMBL8098751

CNC(=O)Nc1ccc(-c2nc(N)cc(C3(S(=O)(=O)c4ccccc4Cl)CC3)n2)cc1

nearest known ligand 0.40

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MTOR P42345 6/20 0.40
PIK3CA P42336 4/20 0.40
PIK3CG P48736 3/20 0.40
CDK1 P06493 3/20 0.37
CDK2 P24941 3/20 0.37
CA12 O43570 1/20 0.37
CA1 P00915 1/20 0.37
CA2 P00918 1/20 0.37
CA9 Q16790 1/20 0.37
F10 P00742 1/20 0.36
SGK1 O00141 2/20 0.36
NAMPT P43490 1/20 0.36
PIP4K2A P48426 1/20 0.35
PIP4K2B P78356 1/20 0.35
NR2E3 Q9Y5X4 1/20 0.35
PIK3CD O00329 4/20 0.35
GSK3A P49840 1/20 0.35
GSK3B P49841 1/20 0.35
SMG1 Q96Q15 1/20 0.35
AKT1 P31749 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8090786 0.90 SGK1 (0.37) MTORF10SGK1NAMPTNR2E3
SCHEMBL8094263 0.88 PIK3CA (0.40) MTORPIK3CAPIK3CGCA12CA1
SCHEMBL8090246 0.87 PIK3CA (0.42) MTORPIK3CAPIK3CGCDK1CDK2
SCHEMBL8091790 0.87 NAMPT (0.38) MTORPIK3CAPIK3CGNAMPTPIK3CD
SCHEMBL8096070 0.84 MTOR (0.40) MTORPIK3CAPIK3CGCDK1CDK2
SCHEMBL8097448 0.83 PIK3CA (0.43) MTORPIK3CAPIK3CGPIP4K2APIP4K2B
SCHEMBL8096342 0.83 PIK3CA (0.41) MTORPIK3CAPIK3CGCDK1CDK2
SCHEMBL8091073 0.83 KMT2A (0.37) MTORPIK3CAPIK3CGCDK1CDK2
SCHEMBL8094423 0.83 CA2 (0.43) MTORPIK3CAPIK3CGCA12CA1
SCHEMBL8092637 0.83 KMT2A (0.42) MTORPIK3CAPIK3CGCA12CA1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed