SCHEMBL8099487

SCHEMBL8099487

Nc1cc(C2(S(=O)(=O)c3cc(F)cc(F)c3)CC2)nc(-c2ccc(NC(=O)NC3CCC3)cc2)n1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA12 O43570 1/20 0.42
CA1 P00915 1/20 0.42
CA2 P00918 1/20 0.42
CA9 Q16790 1/20 0.42
RAB9A P51151 7/20 0.42
NPC1 O15118 6/20 0.42
EPHX1 P07099 4/20 0.42
GAA P10253 2/20 0.40
KDR P35968 2/20 0.38
KIT P10721 1/20 0.38
FLT3 P36888 1/20 0.38
SMN1; SMN2 Q16637 3/20 0.38
MEN1 O00255 3/20 0.37
KMT2A Q03164 3/20 0.37
POLB P06746 2/20 0.37
EPHX2 P34913 1/20 0.37
CYP3A4 P08684 1/20 0.37
CYP2D6 P10635 1/20 0.37
CYP2C9 P11712 1/20 0.37
CYP2C19 P33261 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8084833 0.90 CA12 (0.43) CA12CA1CA2CA9RAB9A
SCHEMBL8098812 0.90 NPC1 (0.43) CA12CA1CA2CA9RAB9A
SCHEMBL8098814 0.88 EPHX1 (0.47) CA12CA1CA2CA9RAB9A
SCHEMBL8089917 0.87 PIK3CA (0.39) CA2CA9KMT2A
SCHEMBL8093179 0.86 RAB9A (0.42) CA12CA1CA2CA9RAB9A
SCHEMBL8104053 0.86 CA2 (0.41) CA12CA1CA2CA9CYP3A4
SCHEMBL8099411 0.86 CA12 (0.44) CA12CA1CA2CA9RAB9A
SCHEMBL8097966 0.85 KIF11 (0.37) MEN1KMT2A
SCHEMBL8099405 0.85 EPHX1 (0.42) CA12CA1CA2CA9RAB9A
SCHEMBL8084016 0.84 CA12 (0.41) CA12CA1CA2CA9RAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2009007748-A2 TRISUBSTITUTED PYRIMIDINE DERIVATIVES FOR THE TREATMENT OF PROLIFERATIVE DISEASES ASTRAZENECA AB (SE) 2009-01-15 WO disclosed