SCHEMBL8101367

SCHEMBL8101367

CCCCN1c2ccc(Br)nc2N(CCCC)c2nc(Br)ccc21

nearest known ligand 0.37

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 5/20 0.37
TP53 P04637 1/20 0.37
MAPK1 P28482 1/20 0.37
PTGS1 P23219 3/20 0.34
PTGS2 P35354 3/20 0.34
MGLL Q99685 2/20 0.34
FAAH O00519 1/20 0.34
ALDH2 P05091 1/20 0.34
ALDH3A1 P30838 1/20 0.34
KMT2A Q03164 3/20 0.34
CNR1 P21554 2/20 0.34
MEN1 O00255 2/20 0.34
TSHR P16473 1/20 0.34
CES1 P23141 2/20 0.33
CDC25A P30304 1/20 0.33
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
GRM2 Q14416 1/20 0.33
POLB P06746 1/20 0.33
NPC1 O15118 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8107632 0.89 ADRA2A (0.36) ALDH1A1TP53MAPK1ALDH2ALDH3A1
SCHEMBL8103441 0.73 KDM4E (0.38) ALDH1A1TP53MAPK1PTGS1PTGS2
SCHEMBL8101881 0.70 ALDH1A1 (0.43) ALDH1A1TP53MAPK1ALDH2ALDH3A1
SCHEMBL8101553 0.68 GAA (0.38) ALDH1A1TP53MAPK1KMT2AMEN1
SCHEMBL15644072 0.65 ALDH1A1 (0.59) ALDH1A1TP53MAPK1PTGS1PTGS2
SCHEMBL31314370 0.64 ALDH1A1 (0.44) ALDH1A1TP53KMT2ACNR1MEN1
SCHEMBL8103457 0.64 ALDH1A1 (0.44) ALDH1A1TP53MAPK1ALDH2ALDH3A1
Bromide SCHEMBL2590637 0.63 DRD2 (0.50) ALDH1A1TP53KMT2ACNR1MEN1
SCHEMBL3635173 0.63 CDC25A (0.61) ALDH1A1PTGS1PTGS2MGLLFAAH
SCHEMBL3023529 0.62 CNR1 (0.42) ALDH1A1TP53MAPK1PTGS1PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127369-A 5,10-dihydrodipyrido[2,3-b:2,3-e]pyrazin and 5,10-dihydrodipyrido[2,3-b:3,2-e]pyrazin compounds ADIR ET COMPAGNIE (FR) 2000-10-03 US disclosed