SCHEMBL8102532

SCHEMBL8102532

COC(=O)C(c1ccccc1Cl)c1cc(Cl)ccc1[N+](=O)[O-]

nearest known ligand 0.54

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 3/20 0.54
MAPK1 P28482 2/20 0.43
TSHR P16473 1/20 0.43
TDP1 Q9NUW8 1/20 0.43
LMNA P02545 3/20 0.42
PDE7A Q13946 1/20 0.41
PKM P14618 1/20 0.41
L3MBTL1 Q9Y468 1/20 0.40
APP P05067 1/20 0.40
SMN1; SMN2 Q16637 2/20 0.40
NPC1 O15118 1/20 0.40
RAB9A P51151 1/20 0.40
MAPT P10636 2/20 0.39
FDFT1 P37268 1/20 0.39
CYP3A4 P08684 1/20 0.39
CYP2D6 P10635 1/20 0.39
SLC6A2 P23975 1/20 0.39
SLC6A4 P31645 1/20 0.39
SLC6A3 Q01959 1/20 0.39
KCNH2 Q12809 1/20 0.39

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5801377 0.84 LMNA (0.47) ALDH1A1MAPK1TDP1LMNAMAPT
SCHEMBL23536629 0.81 ALDH1A1 (0.55) ALDH1A1MAPK1LMNAPKMAPP
SCHEMBL7684242 0.80 ALDH1A1 (0.64) ALDH1A1MAPK1TSHRTDP1LMNA
SCHEMBL948375 0.79 ALDH1A1 (0.51) ALDH1A1MAPK1TSHRTDP1LMNA
SCHEMBL8111568 0.77 ALDH1A1 (0.42) ALDH1A1MAPK1TSHRTDP1LMNA
SCHEMBL4850984 0.75 ALDH1A1 (0.47) ALDH1A1MAPK1TSHRTDP1LMNA
SCHEMBL8102722 0.74 TSHR (0.47) ALDH1A1MAPK1TSHRLMNAPDE7A
SCHEMBL8102779 0.73 TSHR (0.49) ALDH1A1MAPK1TSHRLMNAPDE7A
SCHEMBL4308070 0.72 ALDH1A1 (0.46) ALDH1A1MAPK1TSHRTDP1LMNA
SCHEMBL624054 0.72 ALDH1A1 (0.64) ALDH1A1MAPK1TSHRTDP1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0645378-B1 Condensed seven- or eight-membered heterocyclic compounds useful as squalene synthetase inhibitors TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-08-23 EP disclosed
CN-1054380-C Condensed cyclic compounds and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 2000-07-12 CN disclosed
US-5698691-A ANTICHOLESTEROL AGENT; SYNTHETASE INHIBITOR; FUNGICIDE TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1997-12-16 US disclosed
CN-1106397-A Condensed cyclic compounds and their use TAKEDA CHEMICAL INDUSTRIES LTD (JP) 1995-08-09 CN disclosed
EP-0645378-A1 Condensed seven- or eight-membered heterocyclic compounds useful as squalene synthetase inhibitors Takeda Chemical Industries, Ltd. (JP) 1995-03-29 EP disclosed