SCHEMBL8103486

SCHEMBL8103486

O=C(Cl)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)C(F)(F)F.O=C(Cl)C(F)(F)C(F)(F)C(F)(F)C(F)F.O=C(Cl)C(F)(F)C(F)F

nearest known ligand 0.41

Predicted protein targets (top 6)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.41
KDM4E B2RXH2 1/20 0.32
TSHR P16473 1/20 0.32
TDP1 Q9NUW8 1/20 0.32
L3MBTL1 Q9Y468 2/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7733766 0.94 THRB (0.45) THRBKDM4ETSHRTDP1L3MBTL1
SCHEMBL3423677 0.85 TSHR (0.38) THRBKDM4ETSHRTDP1L3MBTL1
SCHEMBL5705237 0.85 TSHR (0.38) THRBKDM4ETSHRTDP1L3MBTL1
SCHEMBL7729495 0.85 TSHR (0.38) THRBKDM4ETSHRTDP1L3MBTL1
SCHEMBL10617895 0.85 TSHR (0.38) THRBKDM4ETSHRTDP1L3MBTL1
SCHEMBL2796672 0.84 KDM4E (0.40) KDM4ETSHRTDP1
SCHEMBL810833 0.80 THRB (0.59) THRB
SCHEMBL10622506 0.80 THRB (0.59) THRB
SCHEMBL3217875 0.80 THRB (0.59) THRB
SCHEMBL810417 0.80 THRB (0.59) THRB

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0973936-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 2000-01-26 EP disclosed
WO-1998057173-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED PHENYLALANINE LIBRARIES ELI LILLY AND COMPANY (US) 1998-12-17 WO disclosed
EP-0880558-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED INDANE LIBRARIES ELI LILLY AND COMPANY (US) 1998-12-02 EP disclosed
WO-1998046786-A1 COMBINATORIAL LIBRARIES OF PEPTIDOMIMETIC AMINOTHIOETHER ACIDS ELI LILLY AND COMPANY (US) 1998-10-22 WO disclosed
WO-1997026300-A1 COMBINATORIAL PROCESS FOR PREPARING SUBSTITUTED INDANE LIBRARIES ELI LILLY AND COMPANY (US) 1997-07-24 WO disclosed