SCHEMBL8104244

SCHEMBL8104244

Cc1ccc(Cn2cnc(CN(CC(=O)Nc3ccc(C(C)C)cc3)c3cccc(C#N)c3)c2)cc1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
THRB P10828 1/20 0.40
RORC P51449 7/20 0.39
ADRB1 P08588 1/20 0.38
ADRB3 P13945 1/20 0.38
POLB P06746 1/20 0.38
MAPT P10636 2/20 0.37
ALDH1A1 P00352 1/20 0.37
PANK3 Q9H999 1/20 0.37
PSMB5 P28074 1/20 0.36
MCHR1 Q99705 1/20 0.36
CACNA1H O95180 1/20 0.36
LMNA P02545 1/20 0.35
TP53 P04637 1/20 0.35
HTT P42858 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8112410 0.94 NLRP3 (0.38) ADRB1ADRB3POLBMAPTALDH1A1
SCHEMBL8118821 0.88 ALDH1A1 (0.40) POLBMAPTALDH1A1PANK3PSMB5
SCHEMBL8113210 0.86 ALDH1A1 (0.41) RORCPOLBMAPTALDH1A1PANK3
Hydrochloric Acid SCHEMBL8105346 0.85 F10 (0.42) THRBADRB1ADRB3POLBMAPT
SCHEMBL8112927 0.84 MCHR1 (0.37) RORCPOLBMAPTALDH1A1PANK3
SCHEMBL8104036 0.80 MCHR1 (0.38) RORCMAPTALDH1A1PANK3PSMB5
SCHEMBL8122191 0.80 POLB (0.56) THRBRORCPOLBMAPTALDH1A1
SCHEMBL28742149 0.79 POLB (0.47) THRBRORCPOLBMAPTALDH1A1
Hydrochloric Acid SCHEMBL8118836 0.79 F10 (0.42) ADRB1ADRB3MAPTLMNATP53
SCHEMBL8118713 0.79 POLB (0.45) RORCPOLBMAPTALDH1A1PSMB5

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1020434-A1 3-AMIDINOANILINE DERIVATIVES, ACTIVATED BLOOD COAGULATION FACTOR X INHIBITORS, AND INTERMEDIATES FOR PRODUCING BOTH Kissei Pharmaceutical Co., Ltd. (JP) 2000-07-19 EP disclosed