SCHEMBL8104481

SCHEMBL8104481

O=C(N[C@H]1CCN(OC(=O)C(F)(F)F)C1)[C@@H]1CCN1C(=O)OCc1ccc([N+](=O)[O-])cc1

nearest known ligand 0.43

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.38
SIGMAR1 Q99720 2/20 0.37
CCR5 P51681 2/20 0.37
CYP3A4 P08684 1/20 0.36
MAPT P10636 1/20 0.36
CYP2C9 P11712 1/20 0.36
TSHR P16473 1/20 0.36
RAB9A P51151 1/20 0.36
TDP1 Q9NUW8 1/20 0.35
CTSK P43235 2/20 0.35
KLK7 P49862 1/20 0.35
EPHX1 P07099 1/20 0.35
DPP8 Q6V1X1 1/20 0.35
DPP9 Q86TI2 1/20 0.35
CTSB P07858 1/20 0.35
CTSS P25774 1/20 0.35
KCNJ1 P48048 1/20 0.35
ATM Q13315 1/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7463529 0.95 TSHR (0.42) CYP3A4MAPTCYP2C9TSHRRAB9A
SCHEMBL8102754 0.94 CTSK (0.42) CYP3A4MAPTCYP2C9TSHRRAB9A
SCHEMBL8108760 0.90 TSHR (0.44) CYP3A4MAPTCYP2C9TSHRRAB9A
SCHEMBL27410866 0.90 TSHR (0.44) CYP3A4MAPTCYP2C9TSHRRAB9A
SCHEMBL8108799 0.88 CCR2 (0.34) CCR2SIGMAR1CCR5TDP1CTSK
SCHEMBL8439868 0.86 EPHX1 (0.45) CCR2SIGMAR1TDP1CTSKEPHX1
SCHEMBL8438723 0.86 EPHX1 (0.45) CCR2SIGMAR1TDP1CTSKEPHX1
SCHEMBL8094828 0.82 ALDH1A1 (0.45) CCR5MAPT
Trifluoroacetic Acid SCHEMBL8104475 0.80 KCNJ1 (0.40) SIGMAR1CCR5CYP3A4MAPTCYP2C9
SCHEMBL8440251 0.79 TSHR (0.46) CYP3A4MAPTCYP2C9TSHRRAB9A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090802-A BACTERICIDE SANKYO COMPANY, LIMITED (JP) 2000-07-18 US disclosed
EP-0882728-A1 1-METHYLCARBAPENEM DERIVATIVES SANKYO COMPANY LIMITED (JP) 1998-12-09 EP disclosed