SCHEMBL8104943

SCHEMBL8104943

COc1ccc(Sc2cc(S(N)(=O)=O)ccc2[N+](=O)[O-])cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA2 P00918 6/20 0.48
CA1 P00915 3/20 0.48
CA9 Q16790 3/20 0.48
CA12 O43570 1/20 0.48
PDE7A Q13946 2/20 0.47
PTGS2 P35354 3/20 0.43
VCAM1 P19320 1/20 0.43
FBP1 P09467 1/20 0.42
ALDH3A1 P30838 1/20 0.41
KDM4E B2RXH2 1/20 0.41
MEN1 O00255 1/20 0.41
MAPT P10636 1/20 0.41
G6PD P11413 1/20 0.41
PKM P14618 1/20 0.41
MAPK1 P28482 1/20 0.41
KMT2A Q03164 1/20 0.41
NPSR1 Q6W5P4 1/20 0.41
RXFP1 Q9HBX9 1/20 0.41
APOBEC3G Q9HC16 1/20 0.41
SLC6A4 P31645 2/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8105352 0.83 CA2 (0.51) CA2CA1CA9CA12PDE7A
SCHEMBL8098834 0.83 PDE7A (0.64) CA2CA1CA9CA12PDE7A
SCHEMBL8105269 0.81 PTGS2 (0.48) CA2CA1CA9CA12PTGS2
SCHEMBL8964795 0.76 SMN1; SMN2 (0.51) PDE7AMEN1MAPTKMT2ASLC6A4
SCHEMBL8092113 0.76 PTGS2 (0.56) CA2CA1CA9CA12PTGS2
SCHEMBL14486355 0.75 TDP1 (0.51) PDE7AKDM4EMEN1MAPTG6PD
SCHEMBL811285 0.75 PDE7A (0.60) PDE7AKDM4EMEN1MAPTG6PD
SCHEMBL8107622 0.74 IDO1 (0.55) CA2CA1CA9CA12PDE7A
SCHEMBL8107818 0.74 ALDH3A1 (0.61) CA2CA1CA9CA12FBP1
SCHEMBL5956007 0.74 MAPT (0.52) PDE7AKDM4EMEN1MAPTG6PD

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848703-B1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2000-09-27 EP disclosed
US-6004948-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; SIDE EFFECT REDUCTION NYCOMED AUSTRIA GMBH (AT) 1999-12-21 US disclosed
EP-0848703-A1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II Nycomed Austria GmbH (AT) 1998-06-24 EP disclosed
WO-1997003953-A1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 1997-02-06 WO disclosed