SCHEMBL8107622

SCHEMBL8107622

NS(=O)(=O)c1ccc([N+](=O)[O-])c(Sc2cccc(Cl)c2)c1

nearest known ligand 0.55

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
IDO1 P14902 1/20 0.55
PDE7A Q13946 9/20 0.53
VCAM1 P19320 1/20 0.50
PDE7B Q9NP56 3/20 0.49
CA2 P00918 3/20 0.48
CA12 O43570 1/20 0.48
CA1 P00915 1/20 0.48
CA9 Q16790 1/20 0.48
USP7 Q93009 1/20 0.46
CA5A P35218 1/20 0.44
ALDH1A1 P00352 1/20 0.44
KMT2A Q03164 2/20 0.43
NPC1 O15118 1/20 0.43
MAPT P10636 1/20 0.43
PKM P14618 1/20 0.43
MAPK1 P28482 1/20 0.43
LMNA P02545 1/20 0.42

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8098834 0.85 PDE7A (0.64) PDE7AVCAM1PDE7BCA2CA12
SCHEMBL8091331 0.81 CA1 (0.49) PDE7ACA2CA12CA1CA9
SCHEMBL28267868 0.79 PDE7A (0.66) IDO1PDE7APDE7BUSP7ALDH1A1
SCHEMBL8107806 0.79 VCAM1 (0.56) PDE7AVCAM1PDE7BCA2CA12
SCHEMBL8105352 0.77 CA2 (0.51) PDE7AVCAM1PDE7BCA2CA12
SCHEMBL8107618 0.75 NR3C1 (0.42) CA2CA12CA1CA9KMT2A
SCHEMBL28405 0.75 PDE7A (0.77) IDO1PDE7APDE7BALDH1A1KMT2A
SCHEMBL8104943 0.74 CA2 (0.48) PDE7AVCAM1CA2CA12CA1
SCHEMBL5955531 0.72 CCR2 (0.47) IDO1PDE7APDE7BUSP7ALDH1A1
SCHEMBL15307419 0.72 PDE7A (0.64) IDO1PDE7APDE7BUSP7ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0848703-B1 DERIVATIVES OF BENZOSULPHONAMIDES AS INHIBITORS OF THE ENZYME CYCLO-OXYGENASE II NYCOMED AUSTRIA GMBH (AT) 2000-09-27 EP disclosed
US-6004948-A NON-STEROIDAL ANTIINFLAMMATORY AGENTS; SIDE EFFECT REDUCTION NYCOMED AUSTRIA GMBH (AT) 1999-12-21 US disclosed