SCHEMBL8104976

SCHEMBL8104976

CNCCOc1ccc(C)c(C2C3CC4CC(C3)CC2(ONC(C)=O)C4)c1

nearest known ligand 0.36

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 3/20 0.36
ALDH1A1 P00352 3/20 0.36
LMNA P02545 2/20 0.36
POLB P06746 1/20 0.34
P2RX7 Q99572 1/20 0.34
NOS3 P29474 1/20 0.33
NOS1 P29475 1/20 0.33
NOS2 P35228 1/20 0.33
ESR1 P03372 1/20 0.33
EPHX2 P34913 3/20 0.32
MMP2 P08253 1/20 0.32
MMP3 P08254 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP3A4 P08684 1/20 0.32
CYP2C9 P11712 1/20 0.32
CYP2C19 P33261 1/20 0.32
HTT P42858 1/20 0.32
CHEK1 O14757 1/20 0.31
HPGD P15428 1/20 0.31
MAPK1 P28482 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8095608 0.97 KDM4E (0.38) KDM4EALDH1A1LMNAPOLBP2RX7
SCHEMBL8104780 0.85 P2RX7 (0.45) ALDH1A1P2RX7EPHX2
SCHEMBL8104812 0.81 HSP90AA1 (0.37) KDM4EALDH1A1P2RX7EPHX2HTT
SCHEMBL6937092 0.69 CNR2 (0.37) P2RX7EPHX2
SCHEMBL7956634 0.68 P2RX7 (0.72) P2RX7EPHX2MAPK1
SCHEMBL7965604 0.65 P2RX7 (0.71) P2RX7EPHX2
SCHEMBL5075726 0.62 DRD2 (0.61) KDM4EALDH1A1LMNACYP1A2CYP3A4
Hydrochloric Acid SCHEMBL21595615 0.61 DRD2 (0.59) KDM4EALDH1A1LMNACYP1A2CYP3A4
Formic Acid SCHEMBL5073493 0.61 DRD2 (0.56) KDM4EALDH1A1LMNAPOLBCYP1A2
SCHEMBL18295382 0.60 HTR1B (0.52) KDM4EALDH1A1LMNAPDK2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1036058-A1 ADAMANTANE DERIVATIVES AstraZeneca UK Limited (GB) 2000-09-20 EP disclosed
WO-1999029660-A1 ADAMANTANE DERIVATIVES ASTRAZENECA UK LIMITED (GB) 1999-06-17 WO disclosed