SCHEMBL8107465

SCHEMBL8107465

COc1ccc(NNC(=O)C(CC(C)C)S(C)(=O)=O)cc1

nearest known ligand 0.47

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ANPEP P15144 2/20 0.47
PTGS2 P35354 3/20 0.45
ALDH1A1 P00352 3/20 0.44
KMT2A Q03164 1/20 0.44
CTSK P43235 3/20 0.42
CTSL P07711 1/20 0.42
CTSS P25774 1/20 0.42
MMP9 P14780 3/20 0.42
SMN1; SMN2 Q16637 2/20 0.42
MMP2 P08253 2/20 0.42
MMP3 P08254 2/20 0.42
KDM4E B2RXH2 1/20 0.42
GAA P10253 1/20 0.42
HTT P42858 1/20 0.42
HPGD P15428 2/20 0.41
MMP13 P45452 1/20 0.41
HSD17B10 Q99714 1/20 0.41
NPC1 O15118 1/20 0.40
CYP1A2 P05177 1/20 0.40
CYP2D6 P10635 1/20 0.40

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8097957 0.83 GAA (0.57) PTGS2ALDH1A1SMN1; SMN2KDM4EGAA
SCHEMBL3634514 0.70 KMT2A (0.49) PTGS2ALDH1A1KMT2ASMN1; SMN2KDM4E
SCHEMBL26503455 0.70 ANPEP (0.62) ANPEPALDH1A1KMT2ASMN1; SMN2HTT
SCHEMBL20984200 0.69 PTGS2 (0.64) PTGS2ALDH1A1KMT2ASMN1; SMN2KDM4E
SCHEMBL425146 0.68 PTGS2 (0.62) PTGS2ALDH1A1SMN1; SMN2KDM4EGAA
SCHEMBL2831390 0.68 PTGS2 (0.67) PTGS2ALDH1A1SMN1; SMN2KDM4EGAA
SCHEMBL7415077 0.68 MMP9 (0.53) MMP9MMP2MMP3HTTMMP13
SCHEMBL11583393 0.68 AAK1 (0.62) ANPEPALDH1A1KMT2AHTT
SCHEMBL14518056 0.67 L3MBTL1 (0.63) PTGS2ALDH1A1KMT2ASMN1; SMN2KDM4E
SCHEMBL4028705 0.67 PTGS2 (0.60) PTGS2ALDH1A1KMT2ASMN1; SMN2KDM4E

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0993442-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 2000-04-19 EP disclosed
WO-1999001428-A1 HYDRAZINE DERIVATIVES F. HOFFMANN-LA ROCHE AG (CH) 1999-01-14 WO disclosed