SCHEMBL8107544

SCHEMBL8107544

CCCCN1c2ncccc2N(CCCC)c2c(SC)ccnc21

nearest known ligand 0.33

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.33
TP53 P04637 1/20 0.33
MAPK1 P28482 1/20 0.33
ADRA2A P08913 1/20 0.33
ADRA2B P18089 1/20 0.33
ADRA2C P18825 1/20 0.33
ALDH2 P05091 1/20 0.33
ALDH3A1 P30838 1/20 0.33
CES1 P23141 2/20 0.32
CDC25A P30304 1/20 0.32
MEN1 O00255 1/20 0.32
KMT2A Q03164 1/20 0.32
CYP1A2 P05177 1/20 0.32
CYP2D6 P10635 1/20 0.32
CFTR P13569 1/20 0.31
CHRM2 P08172 1/20 0.31
MAPT P10636 1/20 0.30
KDM1A O60341 1/20 0.30
HTT P42858 1/20 0.30

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8101881 0.82 ALDH1A1 (0.43) ALDH1A1TP53MAPK1ADRA2AADRA2B
SCHEMBL8103457 0.80 ALDH1A1 (0.44) ALDH1A1TP53MAPK1ADRA2AADRA2B
SCHEMBL8107632 0.71 ADRA2A (0.36) ALDH1A1TP53MAPK1ADRA2AADRA2B
SCHEMBL8101458 0.71 GRM5 (0.33)
SCHEMBL4316094 0.70 ADRA2A (0.51) ADRA2AADRA2BADRA2CMEN1KMT2A
SCHEMBL8107425 0.70 ADRA2A (0.51) ADRA2AADRA2BADRA2CMEN1KMT2A
SCHEMBL8101315 0.68 ALDH1A1 (0.38) ALDH1A1TP53MAPK1ADRA2AADRA2B
SCHEMBL8093549 0.67 BRD4 (0.39) ALDH1A1ADRA2AADRA2BADRA2CMEN1
SCHEMBL4321443 0.67
SCHEMBL8101460 0.67 PKM (0.36) ALDH1A1TP53MAPK1ALDH2ALDH3A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6127369-A 5,10-dihydrodipyrido[2,3-b:2,3-e]pyrazin and 5,10-dihydrodipyrido[2,3-b:3,2-e]pyrazin compounds ADIR ET COMPAGNIE (FR) 2000-10-03 US disclosed