SCHEMBL8109680

SCHEMBL8109680

CNCCCCc1ccc2c(c1)[S+]([O-])CN2C

nearest known ligand 0.41

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
L3MBTL1 Q9Y468 1/20 0.41
SIGMAR1 Q99720 1/20 0.40
MEN1 O00255 2/20 0.34
KMT2A Q03164 2/20 0.34
CYP1A2 P05177 2/20 0.33
NFKB1 P19838 2/20 0.33
MAPK1 P28482 2/20 0.33
THPO P40225 2/20 0.33
MAPT P10636 2/20 0.33
TP53 P04637 1/20 0.33
ALOX15 P16050 1/20 0.33
TSHR P16473 1/20 0.33
HIF1A Q16665 1/20 0.33
HSD17B10 Q99714 1/20 0.33
DRD2 P14416 2/20 0.32
HTR2A P28223 2/20 0.32
HTR2C P28335 2/20 0.32
DRD3 P35462 2/20 0.32
CYP3A4 P08684 2/20 0.32
SLC6A2 P23975 2/20 0.32

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8871371 0.99 L3MBTL1 (0.40) L3MBTL1SIGMAR1MEN1KMT2ACYP1A2
SCHEMBL8109679 0.90 MAPT (0.41) SIGMAR1CYP1A2NFKB1MAPK1THPO
Hydrochloric Acid SCHEMBL8870609 0.89 MAPT (0.43) SIGMAR1CYP1A2NFKB1MAPK1THPO
SCHEMBL9684037 0.85 S1PR1 (0.38) SIGMAR1TP53HIF1AHSD17B10DRD2
SCHEMBL9684946 0.83 BCHE (0.37) ALOX15
SCHEMBL9437752 0.83 THRA (0.31)
SCHEMBL9685609 0.83 DRD2 (0.39) SIGMAR1CYP1A2MAPK1DRD2HTR2A
Hydrochloric Acid SCHEMBL8870829 0.82 TLR8 (0.35) SIGMAR1CYP1A2HTR2ACYP2D6HRH1
SCHEMBL7760492 0.82
SCHEMBL8110040 0.80 ALDH1A1 (0.39) MEN1KMT2ADRD2SMN1; SMN2ALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 10 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673933-B1 Aminoalkyl benzoxazolinones and benzothiazolinones process for their preparation and compositions containing them ADIR (FR) 2000-11-08 EP disclosed
CN-1055924-C Novel aminoalkyl benzoxazolinones and benzothiazolinones process for their preparation and the pharmaceutical compositions which contain them ADIR (FR) 2000-08-30 CN disclosed
US-5688820-A NERVOUS SYSTEM DISORDERS; PSYCHOLOGICAL DISORDERS ADIR ET COMPAGNIE (FR) 1997-11-18 US disclosed
US-5688811-A PSYCHOLOGICAL DISORDERS; NERVOUS SYSTEM DISORDERS ADIR ET COMPAGNIE (FR) 1997-11-18 US disclosed
US-5534511-A AFFINITY FOR SIGMA RECEPTORS, ANTIINFLAMMATORY, TREATMENT OF ARTHRITIS ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
CN-1112114-A Novel aminoalkyl benzoxazolinones and benzothiazolinones process for their preparation and the pharmaceutical compositions which contain them ADIR (FR) 1995-11-22 CN disclosed
EP-0673933-A1 Aminoalkyl benzoxazolinones and benzothiazolinones process for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1995-09-27 EP disclosed
US-5296477-A Antidepressants ADIR ET COMPAGNIE (FR) 1994-03-22 US disclosed
US-5268381-A Antidepressant or anxiolytic compound ADIR ET COMPAGNIE (FR) 1993-12-07 US disclosed
US-5196434-A Antidepressants, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-03-23 US disclosed