SCHEMBL8114166

SCHEMBL8114166

CN1C[S+]([O-])c2cc(CCCCN)ccc21

nearest known ligand 0.41

Predicted protein targets (top 8)

geneUniProtsupporting neighboursconfidence
TLR8 Q9NR97 6/20 0.36
MAOA P21397 1/20 0.35
SIGMAR1 Q99720 2/20 0.34
CYP1A2 P05177 1/20 0.33
CYP2D6 P10635 1/20 0.33
CYP2C19 P33261 1/20 0.33
HRH1 P35367 2/20 0.33
HTR2A P28223 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8870829 0.99 TLR8 (0.35) TLR8MAOASIGMAR1CYP1A2CYP2D6
SCHEMBL8114240 0.90 KDM4E (0.37) CYP1A2CYP2D6
Hydrochloric Acid SCHEMBL8871802 0.88 LMNA (0.38) CYP1A2CYP2D6
SCHEMBL9684037 0.87 S1PR1 (0.38) SIGMAR1HTR2A
SCHEMBL9437775 0.86 SIGMAR1 (0.36) SIGMAR1CYP1A2CYP2D6
SCHEMBL9684946 0.86 BCHE (0.37)
SCHEMBL9437752 0.86 THRA (0.31)
SCHEMBL9685609 0.85 DRD2 (0.39) SIGMAR1CYP1A2CYP2D6CYP2C19HTR2A
SCHEMBL9437753 0.84 SIGMAR1 (0.39) SIGMAR1CYP1A2CYP2D6
SCHEMBL7760492 0.84

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 7 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0673933-B1 Aminoalkyl benzoxazolinones and benzothiazolinones process for their preparation and compositions containing them ADIR (FR) 2000-11-08 EP disclosed
US-5534511-A AFFINITY FOR SIGMA RECEPTORS, ANTIINFLAMMATORY, TREATMENT OF ARTHRITIS ADIR ET COMPAGNIE (FR) 1996-07-09 US disclosed
EP-0673933-A1 Aminoalkyl benzoxazolinones and benzothiazolinones process for their preparation and compositions containing them ADIR ET COMPAGNIE (FR) 1995-09-27 EP disclosed
US-5296477-A Antidepressants ADIR ET COMPAGNIE (FR) 1994-03-22 US disclosed
US-5268381-A Antidepressant or anxiolytic compound ADIR ET COMPAGNIE (FR) 1993-12-07 US disclosed
US-5196434-A Antidepressants, anxiolytic agents ADIR ET COMPAGNIE (FR) 1993-03-23 US disclosed
EP-0478446-A1 Heterocyclic alkylamines, process for their preparation and pharmaceutical compositions containing them ADIR ET COMPAGNIE (FR) 1992-04-01 EP disclosed