SCHEMBL8124258

SCHEMBL8124258

COc1cc(CO[PH](=O)O)on1

nearest known ligand 0.40

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CHRM1 P11229 4/20 0.40
ALDH1A1 P00352 2/20 0.36
NPC1 O15118 4/20 0.35
RAB9A P51151 4/20 0.35
L3MBTL1 Q9Y468 3/20 0.35
SMN1; SMN2 Q16637 3/20 0.35
POLB P06746 1/20 0.35
KMT2A Q03164 2/20 0.34
MEN1 O00255 1/20 0.34
MAPT P10636 2/20 0.34
TDP1 Q9NUW8 1/20 0.34
MRGPRX4 Q96LA9 1/20 0.34
MAPK1 P28482 1/20 0.33
HSD17B10 Q99714 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8116548 0.87 CHRM1 (0.41) CHRM1ALDH1A1NPC1RAB9AL3MBTL1
SCHEMBL8124187 0.79 ALDH1A1 (0.33) ALDH1A1NPC1RAB9AKMT2AMEN1
SCHEMBL8911503 0.77 CHRM1 (0.40) CHRM1ALDH1A1NPC1RAB9AL3MBTL1
SCHEMBL8123162 0.76 DAO (0.34) ALDH1A1NPC1RAB9AKMT2AMEN1
SCHEMBL8911499 0.73 CHRM1 (0.41) CHRM1NPC1RAB9AL3MBTL1SMN1; SMN2
SCHEMBL3154694 0.73
SCHEMBL8910100 0.73 MMP13 (0.32) ALDH1A1KMT2AMEN1HSD17B10
SCHEMBL11374447 0.71 PTGS1 (0.42) ALDH1A1SMN1; SMN2MAPTTDP1HSD17B10
SCHEMBL10283737 0.71
Phosphonic Acid SCHEMBL8116540 0.70 RAB9A (0.43) ALDH1A1NPC1RAB9AL3MBTL1SMN1; SMN2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 5 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0691962-B1 1-AMINO-3-PHENOXY PROPANE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE BASF AG (DE) 2000-09-13 EP disclosed
US-5675008-A Excitatory amino acid receptor antagonists ELI LILLY AND COMPANY (US) 1997-10-07 US disclosed
US-5670516-A NERVOUS SYSTEM DISORDERS ELI LILLY AND COMPANY (US) 1997-09-23 US disclosed
US-5622953-A DRUG RESISTANT TO ANTICANCER CHEMOTHERAPEUTIC DRUG BASF AKTIENGESELLSCHAFT (DE) 1997-04-22 US disclosed
EP-0691962-A1 1-AMINO-3-PHENOXY PROPANE DERIVATIVES AS MODULATORS OF MULTI-DRUG RESISTANCE BASF AKTIENGESELLSCHAFT (DE) 1996-01-17 EP disclosed