SCHEMBL8130656

SCHEMBL8130656

Brc1ccc(Oc2[c]c3ccccc3cc2)cc1

nearest known ligand 0.39

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CYP2A6 P11509 1/20 0.39
MAPT P10636 1/20 0.37
ABCG2 Q9UNQ0 1/20 0.35
SLC6A2 P23975 2/20 0.34
SLC6A4 P31645 2/20 0.34
SLC6A3 Q01959 1/20 0.34
CES2 O00748 1/20 0.34
CES1 P23141 1/20 0.34
MCL1 Q07820 2/20 0.33
ALDH1A1 P00352 1/20 0.33
TSHR P16473 1/20 0.33
LTA4H P09960 1/20 0.32
CA2 P00918 1/20 0.31
MMP2 P08253 1/20 0.31
MMP9 P14780 1/20 0.31
MMP8 P22894 1/20 0.31
MMP14 P50281 1/20 0.31
CA9 Q16790 1/20 0.31
CA14 Q9ULX7 1/20 0.31
LMNA P02545 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL328780 0.85 LTA4H (0.42) MAPTALDH1A1TSHRLTA4HCA2
SCHEMBL20524986 0.81 CYP2A6 (0.32) CYP2A6ALDH1A1TSHRTDP1
SCHEMBL8125384 0.79
SCHEMBL3237917 0.74 CA1 (0.30) CA2
SCHEMBL8124707 0.72 LMNA (0.46) ALDH1A1LTA4HLMNASMN1; SMN2TDP1
SCHEMBL328940 0.71 LTA4H (0.39) CYP2A6MAPTALDH1A1TSHRLTA4H
SCHEMBL4720994 0.70 RAB9A (0.38) MAPTALDH1A1TSHRMMP2MMP9
SCHEMBL705487 0.70
SCHEMBL64917 0.70 CYP1A2 (0.40) CYP2A6MAPTALDH1A1CA2CA9
SCHEMBL8533924 0.70

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-1028945-A1 SUBSTITUTED PYRIDINE COMPOUNDS AS ANTI-INFLAMMATORY AGENTS Amgen Inc. (US) 2000-08-23 EP disclosed
WO-1999024404-A1 SUBSTITUTED PYRIDINE COMPOUNDS AS ANTI-INFLAMMATORY AGENTS AMGEN INC. (US) 1999-05-20 WO disclosed