SCHEMBL8138192

SCHEMBL8138192

NCC(C(=O)Nc1cc(C(=O)OCc2ccccc2)ccc1Cl)c1ccccc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ROCK2 O75116 4/20 0.50
RAB9A P51151 3/20 0.47
CYP1A2 P05177 1/20 0.47
ALDH1A1 P00352 5/20 0.46
SMN1; SMN2 Q16637 3/20 0.46
HPGD P15428 1/20 0.46
KCNQ2 O43526 1/20 0.46
NPC1 O15118 2/20 0.45
LMNA P02545 2/20 0.45
MAPT P10636 1/20 0.45
KMT2A Q03164 4/20 0.44
MEN1 O00255 3/20 0.44
GAA P10253 1/20 0.44
HDAC1 Q13547 1/20 0.44
HDAC8 Q9BY41 1/20 0.44
HDAC6 Q9UBN7 1/20 0.44
MAPK1 P28482 1/20 0.43
HTT P42858 1/20 0.43
L3MBTL1 Q9Y468 1/20 0.43
SLC6A2 P23975 1/20 0.43

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8135408 0.88 ROCK2 (0.51) ROCK2RAB9AALDH1A1SMN1; SMN2HPGD
SCHEMBL8134584 0.87 ROCK2 (0.50) ROCK2RAB9AALDH1A1SMN1; SMN2NPC1
SCHEMBL8129497 0.85 ALDH1A1 (0.53) ROCK2RAB9AALDH1A1SMN1; SMN2NPC1
SCHEMBL7096106 0.83 ROCK2 (0.59) ROCK2RAB9AKMT2AGAASLC6A2
SCHEMBL8138188 0.83 LNPEP (0.57) ROCK2RAB9ACYP1A2ALDH1A1SMN1; SMN2
SCHEMBL8135411 0.81 RAB9A (0.63) ROCK2RAB9AALDH1A1KMT2AMAPK1
SCHEMBL8133659 0.78 ROCK2 (0.59) ROCK2RAB9ALMNAKMT2ASLC6A2
SCHEMBL9054261 0.77 MAPT (0.57) RAB9ACYP1A2ALDH1A1SMN1; SMN2NPC1
SCHEMBL8122588 0.77 ROCK2 (0.57) ROCK2RAB9AMAPT
SCHEMBL8130076 0.75 ROCK2 (0.51) ROCK2RAB9ACYP1A2MAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0720601-B1 GASTRIN AND CCK RECEPTOR LIGANDS BLACK JAMES FOUNDATION (GB) 2000-10-25 EP disclosed
US-5919829-A Gastrin and cck receptor ligands JAMES BLACK FOUNDATION LIMITED (GB) 1999-07-06 US disclosed
US-5795907-A Gastin and CCK receptor ligands JAMES BLACK FOUNDATION LIMITED (GB) 1998-08-18 US disclosed