SCHEMBL8178641

SCHEMBL8178641

CC(=O)N1CCC(c2nc(COCC(F)(F)F)c(-c3ccccc3)o2)CC1

nearest known ligand 0.49

Predicted protein targets (top 13)

geneUniProtsupporting neighboursconfidence
ADRA1D P25100 1/20 0.49
ADRA1A P35348 1/20 0.49
ADRA1B P35368 1/20 0.49
HCRTR2 O43614 6/20 0.41
HTR2B P41595 1/20 0.40
HDAC3 O15379 1/20 0.40
CYP2C9 P11712 1/20 0.40
HDAC1 Q13547 1/20 0.40
HDAC6 Q9UBN7 1/20 0.40
DGAT1 O75907 1/20 0.39
LMNA P02545 1/20 0.39
KDM1A O60341 1/20 0.38
HCRTR1 O43613 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8166794 0.92 ADRA1D (0.57) ADRA1DADRA1AADRA1BHDAC6LMNA
SCHEMBL8174265 0.85 HCRTR2 (0.42) HCRTR2HTR2BLMNAKDM1AHCRTR1
SCHEMBL8175103 0.81 TRPC3 (0.49) ADRA1DADRA1AADRA1BCYP2C9
SCHEMBL8173512 0.81 HTR2B (0.46) HCRTR2HTR2BLMNAKDM1AHCRTR1
SCHEMBL8180362 0.80 ADRA1D (0.44) ADRA1DADRA1AADRA1BHCRTR2KDM1A
SCHEMBL8174233 0.79 ADRA1D (0.45) ADRA1DADRA1AADRA1BHCRTR2HTR2B
SCHEMBL8166223 0.77 ADRA1D (0.47) ADRA1DADRA1AADRA1BHCRTR2LMNA
SCHEMBL8174942 0.75 ADRA1D (0.45) ADRA1DADRA1AADRA1BCYP2C9
SCHEMBL8174185 0.75 LMNA (0.45) ADRA1DADRA1AADRA1BHTR2BHDAC3
SCHEMBL8166964 0.75 ADRA1D (0.59) ADRA1DADRA1AADRA1BLMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6090825-A Oxazole derivatives as antagonists of alpha 1C andrenergic receptors GLAXO WELLCOME INC. (US) 2000-07-18 US disclosed