SCHEMBL8188366

SCHEMBL8188366

O=S(=O)(CCCO)c1ccc(-c2[nH]nc(Cl)c2-c2ccccc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 17)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.43
HDAC1 Q13547 1/20 0.39
HDAC2 Q92769 1/20 0.39
RPS6KA3 P51812 1/20 0.39
MAPK1 P28482 1/20 0.38
NPSR1 Q6W5P4 1/20 0.38
MMP2 P08253 2/20 0.37
MMP7 P09237 2/20 0.37
MMP14 P50281 2/20 0.37
KEAP1 Q14145 1/20 0.36
NFE2L2 Q16236 1/20 0.36
LOX P28300 1/20 0.34
PTGS2 P35354 3/20 0.34
MMP1 P03956 1/20 0.34
MMP3 P08254 1/20 0.34
MMP9 P14780 1/20 0.34
MMP13 P45452 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8196010 0.92 CA2 (0.43) CA2LOXPTGS2
SCHEMBL8196062 0.89 ALDH1A1 (0.46) CA2PTGS2
SCHEMBL8196926 0.89 CA2 (0.42) CA2LOXPTGS2
SCHEMBL8196195 0.89 PTGS2 (0.40) CA2RPS6KA3MAPK1PTGS2
SCHEMBL8195776 0.84 CA2 (0.41) CA2PTGS2
SCHEMBL8196899 0.83 PTGS2 (0.39) CA2PTGS2
SCHEMBL8200031 0.83 PTGS2 (0.39) CA2PTGS2
SCHEMBL8196142 0.82 PTGS2 (0.37) CA2PTGS2
SCHEMBL8188503 0.82 PTGS2 (0.40) CA2PTGS2
SCHEMBL8188096 0.81 PTGS2 (0.42) PTGS2

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed