SCHEMBL8196010

SCHEMBL8196010

O=S(=O)(CCCO)c1ccc(-c2[nH]nc(Cl)c2-c2ccc(Cl)cc2)cc1

nearest known ligand 0.43

Predicted protein targets (top 12)

geneUniProtsupporting neighboursconfidence
CA2 P00918 2/20 0.43
TBXA2R P21731 1/20 0.39
EDNRB P24530 1/20 0.36
EDNRA P25101 1/20 0.36
PTGS2 P35354 5/20 0.36
PTGS1 P23219 1/20 0.36
PTGDR2 Q9Y5Y4 1/20 0.35
LOX P28300 1/20 0.35
NPC1 O15118 1/20 0.35
KMT2A Q03164 2/20 0.34
LMNA P02545 1/20 0.34
GAA P10253 1/20 0.34

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8195776 0.93 CA2 (0.41) CA2EDNRBEDNRAPTGS2PTGS1
SCHEMBL8188366 0.92 CA2 (0.43) CA2PTGS2LOX
SCHEMBL8196926 0.91 CA2 (0.42) CA2PTGS2PTGS1LOXKMT2A
SCHEMBL8196062 0.91 ALDH1A1 (0.46) CA2PTGS2NPC1KMT2ALMNA
SCHEMBL8196195 0.88 PTGS2 (0.40) CA2TBXA2RPTGS2PTGDR2
SCHEMBL8188503 0.85 PTGS2 (0.40) CA2PTGS2PTGS1PTGDR2
SCHEMBL8196899 0.84 PTGS2 (0.39) CA2PTGS2PTGS1PTGDR2
SCHEMBL8200031 0.84 PTGS2 (0.39) CA2PTGS2PTGS1PTGDR2LMNA
SCHEMBL8196142 0.82 PTGS2 (0.37) CA2PTGS2PTGS1PTGDR2
SCHEMBL8188096 0.82 PTGS2 (0.42) PTGS2PTGS1PTGDR2KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000018741-A2 PYRAZOLE COMPOUNDS AS COX-2 INHIBITORS FUJISAWA PHARMACEUTICAL CO., LTD. (JP) 2000-04-06 WO disclosed