SCHEMBL8200414

SCHEMBL8200414

O=C(Nc1ccccc1-c1ccccc1)c1cccc2c1CCC(CCN1CCC(c3ccccc3)CC1)C2=O

nearest known ligand 0.44

Predicted protein targets (top 9)

geneUniProtsupporting neighboursconfidence
PRCP P42785 1/20 0.44
CHRM3 P20309 15/20 0.43
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
KMT2A Q03164 1/20 0.42
ATM Q13315 1/20 0.42
CCR5 P51681 1/20 0.42
SLC18A3 Q16572 1/20 0.41
HTR2C P28335 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8200188 0.87 KDM4E (0.44) MEN1KMT2ASLC18A3HTR2C
SCHEMBL8203690 0.86 PRCP (0.42) PRCPCCR5SLC18A3HTR2C
SCHEMBL8200402 0.84 HTR2C (0.48) PRCPCHRM3CCR5SLC18A3HTR2C
SCHEMBL8200675 0.84 HTR2C (0.49) PRCPCHRM3MEN1ALDH1A1KMT2A
SCHEMBL8198484 0.83 HTR2C (0.42) MEN1KMT2ASLC18A3HTR2C
SCHEMBL8200595 0.83 ALDH1A1 (0.45) MEN1ALDH1A1KMT2AATMCCR5
SCHEMBL8199345 0.82 CCR2 (0.46) CCR5HTR2C
SCHEMBL8199643 0.82 CCR5 (0.48) PRCPCCR5SLC18A3HTR2C
SCHEMBL8589678 0.82 SIGMAR1 (0.44) MEN1KMT2AHTR2C
SCHEMBL8588349 0.82 SIGMAR1 (0.44) MEN1KMT2AHTR2C

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US claimed
US-6048877-A Tetralone derivatives as antiarrhythmic agents BRISTOL-MYERS SQUIBB COMPANY (US) 2000-04-11 US disclosed
WO-1998036749-A1 TETRALONE DERIVATIVES AS ANTIARRHYTHMIC AGENTS BRISTOL-MYERS SQUIBB COMPANY (US) 1998-08-27 WO disclosed