SCHEMBL8205220

SCHEMBL8205220

CC(C)(C)OC(=O)NCCCc1ccc(C(O)c2cc(Cl)ccc2N)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
CA1 P00915 3/20 0.42
CA2 P00918 3/20 0.42
IDO1 P14902 2/20 0.40
LMNA P02545 1/20 0.40
DRD2 P14416 4/20 0.40
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
BRD4 O60885 1/20 0.38
GAA P10253 1/20 0.38
SIGMAR1 Q99720 1/20 0.38
KDM4E B2RXH2 2/20 0.38
ALDH1A1 P00352 2/20 0.38
HPGD P15428 2/20 0.38
HTT P42858 2/20 0.38
MEN1 O00255 1/20 0.38
KMT2A Q03164 1/20 0.38
SMN1; SMN2 Q16637 1/20 0.38
TP53 P04637 1/20 0.37
GLA P06280 1/20 0.37
MAPT P10636 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6188262 0.94 CA2 (0.44) CA1CA2IDO1LMNADRD2
SCHEMBL8206799 0.89 KDM4E (0.42) CA1CA2IDO1LMNADRD2
SCHEMBL6192309 0.88 GAA (0.48) CA1CA2IDO1LMNAGAA
SCHEMBL6185337 0.83 KDM4E (0.45) CA1CA2IDO1LMNACNR1
SCHEMBL6191215 0.82 AAK1 (0.40) IDO1DRD2GAAKDM4EALDH1A1
SCHEMBL21077910 0.80 DRD2 (0.55) CA1CA2IDO1LMNADRD2
SCHEMBL6190141 0.79 GAA (0.48) CA1CA2IDO1GAAMEN1
SCHEMBL6188694 0.79 CTSL (0.41) IDO1LMNABRD4GAAKDM4E
SCHEMBL6191209 0.78 AAK1 (0.33) IDO1GAAKDM4EALDH1A1HPGD
SCHEMBL22996123 0.78 SMN1; SMN2 (0.54) CA1CA2LMNAGAASIGMAR1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979227-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS Takeda Chemical Industries, Ltd. (JP) 2000-02-16 EP disclosed
WO-1998047882-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-29 WO disclosed