SCHEMBL8206799

SCHEMBL8206799

CC(C)(C)OC(=O)NCCCc1cccc(C(O)c2cc(Cl)ccc2N)c1

nearest known ligand 0.44

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
KDM4E B2RXH2 1/20 0.42
CNR1 P21554 1/20 0.39
CNR2 P34972 1/20 0.39
CTSL P07711 1/20 0.39
IDO1 P14902 2/20 0.39
SIGMAR1 Q99720 2/20 0.38
ALDH1A1 P00352 2/20 0.38
LMNA P02545 1/20 0.38
PKM P14618 1/20 0.38
HPGD P15428 1/20 0.38
TSHR P16473 1/20 0.38
MAPK1 P28482 1/20 0.38
DRD2 P14416 4/20 0.38
MAPT P10636 2/20 0.38
CA1 P00915 1/20 0.38
CA2 P00918 1/20 0.38
ATM Q13315 1/20 0.37
BRD4 O60885 1/20 0.37

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL6185337 0.94 KDM4E (0.45) KDM4ECNR1CTSLIDO1ALDH1A1
SCHEMBL8205220 0.89 CA1 (0.42) KDM4ECNR1CNR2IDO1SIGMAR1
SCHEMBL6188694 0.88 CTSL (0.41) KDM4ECTSLIDO1ALDH1A1LMNA
SCHEMBL6188262 0.83 CA2 (0.44) KDM4EIDO1ALDH1A1LMNAPKM
SCHEMBL28745235 0.83 GAA (0.40) KDM4ECTSLIDO1ALDH1A1LMNA
SCHEMBL7665564 0.82 AAK1 (0.39) KDM4ECTSLIDO1ALDH1A1HPGD
SCHEMBL8210587 0.81 ALDH1A1 (0.39) KDM4EALDH1A1LMNATSHRMAPK1
SCHEMBL6188601 0.81 GLS (0.42) KDM4ECTSLALDH1A1LMNABRD4
SCHEMBL11952529 0.80 KDM4E (0.58) KDM4ECTSLSIGMAR1ALDH1A1LMNA
SCHEMBL8211448 0.80 DHFR (0.36) SIGMAR1MAPTCA1CA2ATM

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0979227-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS Takeda Chemical Industries, Ltd. (JP) 2000-02-16 EP disclosed
WO-1998047882-A1 4,1-BENZOXAZEPINES, THEIR ANALOGUES, AND THEIR USE AS SOMATOSTATIN AGONISTS TAKEDA CHEMICAL INDUSTRIES, LTD. (JP) 1998-10-29 WO disclosed