SCHEMBL8206330

SCHEMBL8206330

COC(=O)c1ccc(C(=O)Nc2sc(Cl)cc2C(=O)NCc2ccccc2)cc1

nearest known ligand 0.50

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MEN1 O00255 1/20 0.50
KMT2A Q03164 1/20 0.50
SMN1; SMN2 Q16637 1/20 0.50
KDM4E B2RXH2 5/20 0.47
SCD O00767 1/20 0.46
CA1 P00915 1/20 0.46
CA2 P00918 1/20 0.46
L3MBTL1 Q9Y468 1/20 0.46
ALDH1A1 P00352 2/20 0.46
PKM P14618 1/20 0.46
HPGD P15428 4/20 0.45
TP53 P04637 2/20 0.45
GLA P06280 1/20 0.45
MAPT P10636 3/20 0.45
PPARG P37231 2/20 0.45
BCL2 P10415 1/20 0.45
MCL1 Q07820 1/20 0.45
MGAM O43451 1/20 0.44
AMY1A P0DUB6 1/20 0.44
HSP90AA1 P07900 1/20 0.44

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8199930 0.89 MGLL (0.52) MEN1KMT2ASMN1; SMN2KDM4EALDH1A1
SCHEMBL8206605 0.89 NPC1 (0.48) MEN1KMT2ASMN1; SMN2KDM4EALDH1A1
SCHEMBL8210425 0.89 EPHX2 (0.51) KMT2ASMN1; SMN2CA1CA2ALDH1A1
SCHEMBL8210714 0.88 KDM4E (0.51) MEN1KMT2ASMN1; SMN2KDM4ESCD
SCHEMBL8212457 0.86 AKR1B1 (0.49) MEN1KMT2ASMN1; SMN2ALDH1A1HPGD
SCHEMBL8212903 0.86 MEN1 (0.49) MEN1KMT2ASMN1; SMN2KDM4ESCD
SCHEMBL8206984 0.86 ALDH1A1 (0.54) MEN1KMT2ASMN1; SMN2KDM4ESCD
SCHEMBL8199066 0.85 LMNA (0.52) MEN1KMT2ASMN1; SMN2HPGDMAPT
SCHEMBL8245383 0.85 ROCK2 (0.52) MEN1KMT2ASMN1; SMN2ALDH1A1HPGD
SCHEMBL8212431 0.82 TDP1 (0.54) MEN1KMT2ASMN1; SMN2KDM4EALDH1A1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143777-A ENZYME INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-07 US disclosed