SCHEMBL8207604

SCHEMBL8207604

Brc1ccc(C[CH]c2ccccc2)cc1

nearest known ligand 0.42

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 0.42
TDP1 Q9NUW8 1/20 0.42
G6PD P11413 1/20 0.41
MAOB P27338 2/20 0.41
MAOA P21397 1/20 0.41
MAPK1 P28482 1/20 0.41
CYP1B1 Q16678 1/20 0.39
GPR52 Q9Y2T5 1/20 0.38
PDPK1 O15530 1/20 0.38
CYP2A6 P11509 1/20 0.37
L3MBTL1 Q9Y468 1/20 0.37
HTR2A P28223 2/20 0.37
TAAR1 Q96RJ0 1/20 0.37
EPHX1 P07099 1/20 0.37
MAPT P10636 2/20 0.36
MEN1 O00255 1/20 0.36
LMNA P02545 1/20 0.36
GAA P10253 1/20 0.36
HPGD P15428 1/20 0.36
RAB9A P51151 1/20 0.36

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8199494 0.91 MAOB (0.46) ALDH1A1TDP1G6PDMAOBMAPK1
SCHEMBL69726 0.84 MAOB (0.57) ALDH1A1MAOBMAOACYP2A6L3MBTL1
SCHEMBL15527347 0.79 MAOB (0.48) ALDH1A1TDP1G6PDMAOBMAOA
SCHEMBL3847991 0.79 MAOB (0.48) ALDH1A1TDP1G6PDMAOBMAOA
SCHEMBL6207299 0.79 MEN1 (0.42) ALDH1A1MEN1LMNAGAAKMT2A
SCHEMBL3241749 0.78 LMNA (0.42) ALDH1A1TDP1MAOBMAOAMAPK1
SCHEMBL4348469 0.78 ESR1 (0.45) TDP1MAOBMAOACYP1B1TAAR1
SCHEMBL8840747 0.78 SIGMAR1 (0.44) ALDH1A1TDP1G6PDMAOBCYP1B1
SCHEMBL5852576 0.78 MAOB (0.52) ALDH1A1TDP1MAOBMAOACYP1B1
SCHEMBL8210813 0.78 NFE2L2 (0.52) ALDH1A1MAOBMAOACYP2A6L3MBTL1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6030975-A ANTAGONIST OF ENDOTHELINS, I.E. INHIBITION OF BINDING WITH RECEPTOR; ANTITUMOR AND -CARCINOGENIC AGENTS; SIDE EFFECT REDUCTION BASF AKTIENGESELLSCHAFT (DE) 2000-02-29 US disclosed
US-5840722-A ADMINISTERING TO INHIBIT ENDOTHELIN RECEPTORS BASF AKTIENGESELLSCHAFT (DE) 1998-11-24 US disclosed
US-5703017-A HERBICIDES, PLANT GROWTH REGULATORS BASF AKTIENGESELLSCHAFT (DE) 1997-12-30 US disclosed
CN-1121711-A 3-(hetero)aryl carboxylic acid derivatives, methods of preparing them and intermediates used in their preparation BASF AG (DE) 1996-05-01 CN disclosed