SCHEMBL8207643

SCHEMBL8207643

COC(=O)c1ccc(C(=O)Nc2sc3c(c2C(=O)NC(Cc2ccccc2)C2=COCO2)CCCC3)cc1

nearest known ligand 0.51

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
MGAM O43451 1/20 0.51
AMY1A P0DUB6 1/20 0.51
GLO1 Q04760 1/20 0.48
TP53 P04637 3/20 0.47
KMT2A Q03164 3/20 0.47
RAB9A P51151 3/20 0.47
ALDH1A1 P00352 2/20 0.47
NPC1 O15118 2/20 0.47
MEN1 O00255 2/20 0.47
MAPT P10636 4/20 0.47
LMNA P02545 2/20 0.47
HPGD P15428 2/20 0.47
KDM4E B2RXH2 1/20 0.47
CYP1A2 P05177 1/20 0.47
CYP3A4 P08684 1/20 0.47
CYP2C9 P11712 1/20 0.47
CYP2C19 P33261 1/20 0.47
KIF11 P52732 1/20 0.47
FLT3 P36888 1/20 0.46
ATM Q13315 1/20 0.46

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7889393 0.92 KMT2A (0.52) MGAMAMY1AGLO1TP53KMT2A
SCHEMBL8206343 0.85 MAPT (0.47) TP53ALDH1A1MAPTHPGDKDM4E
SCHEMBL8208116 0.83 MAPT (0.50) TP53KMT2ARAB9AALDH1A1NPC1
SCHEMBL8200088 0.82 FLT3 (0.44) MGAMAMY1ATP53KMT2ARAB9A
SCHEMBL8206432 0.81 TAAR1 (0.54) TP53KMT2ARAB9AALDH1A1NPC1
SCHEMBL8212434 0.80 SMN1; SMN2 (0.39) KMT2AALDH1A1MEN1MAPTLMNA
SCHEMBL8200396 0.80 ALDH1A1 (0.44) KMT2ARAB9AALDH1A1MEN1MAPT
SCHEMBL8198895 0.79 SMN1; SMN2 (0.38) KMT2ARAB9AALDH1A1NPC1MEN1
SCHEMBL8200375 0.78 ALDH1A1 (0.41) KMT2ARAB9AALDH1A1MEN1MAPT
SCHEMBL8211459 0.78 MGAM (0.77) MGAMAMY1AGLO1TP53KMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-6143777-A ENZYME INHIBITORS MERCK PATENT GESELLSCHAFT MIT BESCHRANKTER HAFTUNG (DE) 2000-11-07 US disclosed