SCHEMBL8210586

SCHEMBL8210586

O=C(O)c1cc2cc(NC(=O)c3ccc(C(=O)Nc4ccc5[nH]c(C(=O)O)cc5c4)o3)ccc2[nH]1

nearest known ligand 0.59

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
SMAD3 P84022 1/20 0.51
NHERF1 O14745 3/20 0.51
NPC1 O15118 4/20 0.50
HPGD P15428 3/20 0.50
KDM4E B2RXH2 3/20 0.50
MAPT P10636 3/20 0.50
KMT2A Q03164 3/20 0.50
RAB9A P51151 3/20 0.50
ALDH1A1 P00352 2/20 0.50
PYGL P06737 2/20 0.50
LMNA P02545 2/20 0.50
HSD17B10 Q99714 2/20 0.50
MEN1 O00255 2/20 0.50
F7 P08709 1/20 0.50
F3 P13726 1/20 0.50
PIN1 Q13526 1/20 0.50
PDPK1 O15530 1/20 0.50
TSHR P16473 1/20 0.50
NFKB1 P19838 1/20 0.50
APEX1 P27695 1/20 0.50

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL3043508 0.88 PTPN1 (0.51) NPC1HPGDKDM4EMAPTKMT2A
SCHEMBL5733671 0.84 RAB9A (0.62) NPC1HPGDKDM4EMAPTKMT2A
SCHEMBL8204182 0.83 NHERF1 (0.60) SMAD3NHERF1NPC1HPGDKDM4E
SCHEMBL3058666 0.82 KDM4E (0.62) NHERF1NPC1HPGDKDM4EMAPT
SCHEMBL7470448 0.82 SMAD3 (0.60) SMAD3NHERF1NPC1HPGDKDM4E
SCHEMBL8197851 0.82 SMAD3 (0.60) SMAD3NHERF1NPC1HPGDKDM4E
SCHEMBL27520204 0.82 NPC1 (0.53) NHERF1NPC1HPGDMAPTKMT2A
SCHEMBL5679468 0.82 FLT3 (0.51) SMAD3NHERF1NPC1HPGDKDM4E
SCHEMBL10466165 0.82 MAOA (0.71) NHERF1NPC1HPGDKDM4EMAPT
SCHEMBL8205569 0.81 MMP13 (0.72) NPC1HPGDKDM4EMAPTKMT2A

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 4 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0359454-B1 CC-1065 analogs having two CPI subunits UPJOHN CO (US) 2000-12-27 EP disclosed
US-5541339-A ANTITUMOR AGENTS THE UPJOHN COMPANY (US) 1996-07-30 US disclosed
WO-1990002746-A1 NOVEL CC-1065 ANALOGS HAVING TWO CPI SUBUNITS THE UPJOHN COMPANY (US) 1990-03-22 WO disclosed
EP-0359454-A1 Novel CC-1065 analogs having two CPI subunits THE UPJOHN COMPANY (US) 1990-03-21 EP disclosed