SCHEMBL8217404

SCHEMBL8217404

CC(C)(C)OC(=O)N(CCc1cccc(F)c1)C1CCCC1

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
PPARG P37231 1/20 0.44
PPARD Q03181 1/20 0.44
PPARA Q07869 1/20 0.44
TAAR1 Q96RJ0 1/20 0.44
OPRM1 P35372 5/20 0.43
NPC1 O15118 1/20 0.43
RAB9A P51151 1/20 0.43
KMT2A Q03164 1/20 0.43
GPR119 Q8TDV5 1/20 0.41
SIGMAR1 Q99720 1/20 0.40
AGER Q15109 2/20 0.40
MTNR1A P48039 1/20 0.40
L3MBTL1 Q9Y468 1/20 0.39
HTR1A P08908 1/20 0.39
SLC6A4 P31645 1/20 0.39
RIPK1 Q13546 1/20 0.39
ADRA2C P18825 1/20 0.38
HRH2 P25021 1/20 0.38
HTR2B P41595 1/20 0.38
SLC6A3 Q01959 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL2258375 0.87 SLC18A3 (0.40) PPARGPPARDPPARATAAR1OPRM1
SCHEMBL1798916 0.86 L3MBTL1 (0.42) PPARGPPARDPPARAOPRM1L3MBTL1
SCHEMBL12363036 0.86 TAAR1 (0.40) PPARGPPARDPPARATAAR1OPRM1
SCHEMBL4525149 0.81 GRM2 (0.40) OPRM1SIGMAR1L3MBTL1
SCHEMBL14191955 0.81 GPR119 (0.37) PPARGPPARDPPARATAAR1OPRM1
Formic Acid SCHEMBL27903276 0.80 L3MBTL1 (0.47) PPARGPPARDPPARAOPRM1KMT2A
SCHEMBL2260853 0.79 ALDH1A1 (0.40) PPARGPPARDPPARAKMT2AGPR119
SCHEMBL5042994 0.79 SLC6A2 (0.53) OPRM1SLC6A4SLC6A3
SCHEMBL4511972 0.78 SIGMAR1 (0.45) NPC1RAB9ASIGMAR1
SCHEMBL2257504 0.78 TAAR1 (0.50) TAAR1KMT2ASIGMAR1HTR1ASLC6A4

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2008042353-A1 POTENT AND HIGHLY SELECTIVE HETEROAROMATIC INHIBITORS OF NEURONAL NITRIC OXIDE SYNTHASE NORTHWESTERN UNIVERSITY (US) 2008-04-10 WO disclosed