SCHEMBL8219938

SCHEMBL8219938

O=Cc1[nH]c2cccc(Cl)c2c1Cl

nearest known ligand 0.44

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ERCC5 P28715 1/20 0.44
FEN1 P39748 1/20 0.44
MEN1 O00255 1/20 0.42
ALDH1A1 P00352 1/20 0.42
KMT2A Q03164 1/20 0.42
TDP1 Q9NUW8 1/20 0.42
GRIN2D O15399 2/20 0.41
GRIN3B O60391 2/20 0.41
GRIN1 Q05586 2/20 0.41
GRIN2A Q12879 2/20 0.41
GRIN2B Q13224 2/20 0.41
GRIN2C Q14957 2/20 0.41
GRIN3A Q8TCU5 2/20 0.41
DYRK1A Q13627 1/20 0.40
CHEK1 O14757 1/20 0.39
GPR17 Q13304 1/20 0.38
PBRM1 Q86U86 1/20 0.38
GPR84 Q9NQS5 1/20 0.37
GAA P10253 1/20 0.37
PSMB8 P28062 2/20 0.35

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL5666588 0.78 CA12 (0.44) MEN1ALDH1A1KMT2ATDP1GRIN2D
SCHEMBL31619545 0.75 ERCC5 (0.53) ERCC5FEN1GRIN2DGRIN3BGRIN1
SCHEMBL6009055 0.75 ERCC5 (0.53) ERCC5FEN1GRIN2DGRIN3BGRIN1
SCHEMBL29954948 0.74 MEN1 (0.52) ERCC5FEN1MEN1ALDH1A1KMT2A
SCHEMBL10464296 0.74 DYRK1A (0.46) ERCC5FEN1GRIN2DGRIN3BGRIN1
SCHEMBL1336656 0.73 KIF11 (0.46) MEN1ALDH1A1KMT2AGAA
SCHEMBL29953769 0.73 KIF11 (0.46) MEN1ALDH1A1KMT2AGAA
SCHEMBL7493525 0.71 ALDH1A1 (0.48) ERCC5FEN1MEN1ALDH1A1KMT2A
SCHEMBL20276479 0.71 ERCC5 (0.50) ERCC5FEN1GRIN2DGRIN3BGRIN1
SCHEMBL9038402 0.69 GPR17 (0.61) ERCC5FEN1ALDH1A1GRIN2DGRIN3B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2000071524-A1 2-NH-PYRIDONES AND PYRIMIDONES AS MRS INHIBITORS SMITHKLINE BEECHAM PLC (GB) 2000-11-30 WO disclosed