SCHEMBL8249388

SCHEMBL8249388

CC(C)(C)OC(=O)NCc1ccc(Br)c(O)c1

nearest known ligand 0.49

Predicted protein targets (top 19)

geneUniProtsupporting neighboursconfidence
HDAC1 Q13547 2/20 0.48
CA1 P00915 3/20 0.47
CA2 P00918 3/20 0.47
L3MBTL1 Q9Y468 1/20 0.46
NAMPT P43490 2/20 0.44
GAA P10253 1/20 0.44
KDM4A O75164 1/20 0.44
TSHR P16473 1/20 0.43
CA12 O43570 2/20 0.43
CA9 Q16790 2/20 0.43
FPR3 P25089 1/20 0.43
FPR2 P25090 1/20 0.43
GRM2 Q14416 1/20 0.43
GLS O94925 1/20 0.42
ERCC1 P07992 1/20 0.42
ERCC4 Q92889 1/20 0.42
HDAC10 Q969S8 1/20 0.42
HDAC6 Q9UBN7 1/20 0.42
HPN P05981 1/20 0.41

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL1985433 0.89 HDAC1 (0.51) HDAC1CA1CA2L3MBTL1NAMPT
SCHEMBL5749285 0.87 ERCC1 (0.56) HDAC1CA1CA2L3MBTL1NAMPT
SCHEMBL850268 0.86 MEN1 (0.47) HDAC1CA1CA2L3MBTL1NAMPT
SCHEMBL508353 0.84 TSHR (0.56) HDAC1CA1CA2L3MBTL1NAMPT
SCHEMBL507617 0.84 GRM2 (0.47) HDAC1CA1CA2L3MBTL1NAMPT
SCHEMBL31142951 0.84 ALDH1A1 (0.48) HDAC1CA1CA2L3MBTL1NAMPT
SCHEMBL24838807 0.83 ALDH1A1 (0.51) L3MBTL1TSHRGRM2
SCHEMBL14450526 0.83 GRM2 (0.48) HDAC1CA1CA2L3MBTL1NAMPT
SCHEMBL31431581 0.83 HDAC1 (0.48) HDAC1CA1CA2L3MBTL1NAMPT
SCHEMBL3688009 0.83 HDAC1 (0.48) HDAC1CA1CA2L3MBTL1NAMPT

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 14 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-4688750-A1 SUBSTITUTED INDAZOLE PROPIONIC ACID DERIVATIVE COMPOUNDS AND USES THEREOF AS AMPK ACTIVATORS Pfizer Inc. (US) 2026-02-11 EP disclosed
WO-2024209363-A1 SUBSTITUTED INDAZOLE PROPIONIC ACID DERIVATIVE COMPOUNDS AND USES THEREOF AS AMPK ACTIVATORS PFIZER INC. (US) 2024-10-10 WO disclosed
US-20240336572-A1 SUBSTITUTED INDAZOLE PROPIONIC ACID DERIVATIVE COMPOUNDS AND USES THEREOF PFIZER INC. (US) 2024-10-10 US disclosed
US-20120015920-A1 HETEROBICYCLIC METALLOPROTEASE INHIBITORS ALANTOS PHARMACEUTICALS HOLDING, INC. (US) 2012-01-19 US disclosed
US-20120015920-A1 HETEROBICYCLIC METALLOPROTEASE INHIBITORS ALANTOS PHARMACEUTICALS HOLDING, INC. (US) 2012-01-19 US disclosed
US-7795245-B2 Heterobicyclic metalloprotease inhibitors Atlantos Pharmaceuticals Holding, Inc. (US) 2010-09-14 US disclosed
US-7795245-B2 Heterobicyclic metalloprotease inhibitors Atlantos Pharmaceuticals Holding, Inc. (US) 2010-09-14 US disclosed
US-20090312312-A1 Heterobicyclic Metalloprotease Inhibitors ALANTOS PHARMACEUTICALS HOLDING, INC. (US) 2009-12-17 US disclosed
US-20090312312-A1 Heterobicyclic Metalloprotease Inhibitors ALANTOS PHARMACEUTICALS HOLDING, INC. (US) 2009-12-17 US disclosed
US-20090137547-A1 Heterobicyclic metalloprotease inhibitors ALANTOS PHARMACEUTICALS HOLDING, INC. 2009-05-28 US disclosed
US-20090137547-A1 Heterobicyclic metalloprotease inhibitors ALANTOS PHARMACEUTICALS HOLDING, INC. 2009-05-28 US disclosed
US-20070155738-A1 Heterobicyclic metalloprotease inhibitors ALANTOS PHARMACEUTICALS, INC. 2007-07-05 US disclosed
US-20070155738-A1 Heterobicyclic metalloprotease inhibitors ALANTOS PHARMACEUTICALS, INC. 2007-07-05 US disclosed
WO-2006128184-A2 PYRIMIDINE OR TRIAZINE FUSED BICYCLIC METALLOPROTEASE INHIBITORS ALANTOS-PHARMACEUTICALS, INC. (US) 2006-11-30 WO disclosed

Patent text — is the patent's own abstract consistent with the prediction?

For each of this compound's patents that has machine-readable text (5 of them — usually the abstract, not the full specification), we ask MedCPT which protein the text reads most about, and where the chemistry-predicted target lands among 4885 human targets. A high rank means the patent's own wording is consistent with the prediction — a weak, independent signal, not proof of activity.

PatentTitleText reads most aboutPredicted target · text-rank
US-20240336572-A1 SUBSTITUTED INDAZOLE PROPIONIC ACID DERIVATIVE COMPOUNDS AND USES THEREOF PRKAG3, PRKAG1, PRKAG2 HDAC1 1175/4885CA1 4045/4885CA2 1419/4885
US-20090312312-A1 Heterobicyclic Metalloprotease Inhibitors MMP13, TIMP3, MMP3 HDAC1 104/4885CA1 350/4885CA2 196/4885
US-20120015920-A1 HETEROBICYCLIC METALLOPROTEASE INHIBITORS MMP13, TIMP3, MMP3 HDAC1 104/4885CA1 350/4885CA2 196/4885
US-20090137547-A1 Heterobicyclic metalloprotease inhibitors MMP13, TIMP3, MMP3 HDAC1 104/4885CA1 350/4885CA2 196/4885
US-20070155738-A1 Heterobicyclic metalloprotease inhibitors MMP13, TIMP3, MMP3 HDAC1 104/4885CA1 350/4885CA2 196/4885

“Text reads most about” is the patent abstract's nearest protein in MedCPT space (background-debiased). Only ~1.4% of patents have machine-readable text, so most compounds won't have this panel.