SCHEMBL8264342

SCHEMBL8264342

O=C(O)Cn1cc(CNC2CC2)c2ccccc21

nearest known ligand 0.54

Predicted protein targets (top 15)

geneUniProtsupporting neighboursconfidence
KMT2A Q03164 2/20 0.52
ALDH1A1 P00352 6/20 0.50
TBXAS1 P24557 1/20 0.50
STAT3 P40763 1/20 0.49
S1PR2 O95136 1/20 0.48
MCL1 Q07820 1/20 0.47
KDM4E B2RXH2 4/20 0.47
MAPT P10636 1/20 0.47
GFER P55789 1/20 0.47
TSHR P16473 1/20 0.46
RXFP1 Q9HBX9 1/20 0.46
HPGD P15428 1/20 0.46
PTGDR2 Q9Y5Y4 1/20 0.46
SMN1; SMN2 Q16637 1/20 0.46
ALOX5 P09917 1/20 0.45

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL10183497 0.83 LMNA (0.58) KMT2AALDH1A1KDM4EMAPTTSHR
SCHEMBL8264846 0.82 GAA (0.44) KMT2AALDH1A1KDM4ESMN1; SMN2
SCHEMBL1518291 0.81 HTR2C (0.54) KMT2AALDH1A1TSHRSMN1; SMN2
SCHEMBL8264241 0.81 P2RX7 (0.46) KMT2A
SCHEMBL1518225 0.81 PDE4B (0.42) KMT2AALDH1A1KDM4EMAPTHPGD
SCHEMBL30979650 0.81 ALDH1A1 (0.55) KMT2AALDH1A1TBXAS1STAT3S1PR2
SCHEMBL8264949 0.80 ICMT (0.51) KMT2AALDH1A1KDM4EMAPTRXFP1
SCHEMBL1074732 0.79 MAPK1 (0.47) KMT2AALDH1A1KDM4EHPGDSMN1; SMN2
SCHEMBL8263899 0.79 CNR1 (0.46)
SCHEMBL27854488 0.78 DNM2 (0.46) TSHR

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 1 patent. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
WO-2006074924-A1 3,4,(5)-SUBSTITUTED TETRAHVDROPYRIDINES NOVARTIS AG (CH) 2006-07-20 WO disclosed