SCHEMBL8275407

SCHEMBL8275407

CC(=O)c1ccc(NS(=O)(=O)c2ccc3ccccc3c2)cc1

nearest known ligand 1.00 ✓ in ChEMBL — recovers established targets

Predicted protein targets (top 20)

geneUniProtsupporting neighboursconfidence
ALDH1A1 P00352 4/20 1.00
SMN1; SMN2 Q16637 3/20 1.00
GAA P10253 2/20 1.00
LMNA P02545 2/20 1.00
HDAC1 Q13547 2/20 0.71
HDAC3 O15379 1/20 0.71
HDAC4 P56524 1/20 0.71
HDAC7 Q8WUI4 1/20 0.71
HDAC2 Q92769 1/20 0.71
HDAC10 Q969S8 1/20 0.71
HDAC11 Q96DB2 1/20 0.71
HDAC8 Q9BY41 1/20 0.71
HDAC6 Q9UBN7 1/20 0.71
HDAC9 Q9UKV0 1/20 0.71
HDAC5 Q9UQL6 1/20 0.71
PLAU P00749 2/20 0.70
ATM Q13315 1/20 0.69
CA12 O43570 1/20 0.68
CA9 Q16790 1/20 0.68
MAPT P10636 5/20 0.64

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL7782154 0.87 ALDH1A1 (0.77) ALDH1A1SMN1; SMN2GAALMNAHDAC1
SCHEMBL15480550 0.84 LMNA (0.73) ALDH1A1SMN1; SMN2GAALMNAHDAC1
SCHEMBL8277295 0.83 HDAC3 (1.00) ALDH1A1SMN1; SMN2GAALMNAHDAC1
SCHEMBL8276342 0.82 HDAC1 (0.70) ALDH1A1SMN1; SMN2GAALMNAHDAC1
SCHEMBL808105 0.82 ATM (0.72) ALDH1A1SMN1; SMN2GAALMNAHDAC1
SCHEMBL7791354 0.82 PLAU (0.72) ALDH1A1SMN1; SMN2GAALMNAHDAC1
SCHEMBL17913100 0.82 CA12 (1.00) ALDH1A1SMN1; SMN2GAALMNACA12
SCHEMBL2201204 0.82 CA12 (0.87) ALDH1A1SMN1; SMN2GAALMNAHDAC1
SCHEMBL20021987 0.81 PGR (0.77) ALDH1A1SMN1; SMN2GAALMNAHDAC1
SCHEMBL28396503 0.81 PGR (0.77) ALDH1A1SMN1; SMN2GAALMNAHDAC1

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
US-7470722-B2 Multicyclic sulfonamide compounds as inhibitors of histone deacetylase for the treatment of disease KALYPSYS, INC. (US) 2008-12-30 US disclosed
US-7470722-B2 Multicyclic sulfonamide compounds as inhibitors of histone deacetylase for the treatment of disease KALYPSYS, INC. (US) 2008-12-30 US disclosed
WO-2005123089-A2 MULTICYCLIC SULFONAMIDE COMPOUNDS AS INHIBITORS OF HISTONE DEACETYLASE FOR THE TREATMENT OF DISEASE KALYPSYS, INC. (US) 2005-12-29 WO disclosed