SCHEMBL8300207

SCHEMBL8300207

COC(C(=O)O)C1CCC(N2CCC(CCNc3ccnnc3)CC2)CC1

nearest known ligand 0.34

Predicted protein targets (top 14)

geneUniProtsupporting neighboursconfidence
CCR2 P41597 1/20 0.34
RAB9A P51151 1/20 0.34
LRRK2 Q5S007 5/20 0.34
BDKRB1 P46663 3/20 0.33
GRIN2B Q13224 1/20 0.32
OPRM1 P35372 1/20 0.32
OPRL1 P41146 1/20 0.32
CHRM4 P08173 1/20 0.32
CCR3 P51677 1/20 0.32
CCRL2 O00421 1/20 0.32
CHRM2 P08172 1/20 0.31
CXCR3 P49682 1/20 0.31
GPR119 Q8TDV5 1/20 0.31
BCHE P06276 1/20 0.31

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8305658 0.81 CCNT1 (0.38) LRRK2GRIN2BCHRM4CXCR3
SCHEMBL8792322 0.78 BDKRB1 (0.31) CCR2BDKRB1GRIN2BGPR119
SCHEMBL8617208 0.76 KDM4E (0.40) GRIN2B
SCHEMBL8301158 0.76 CCR2 (0.35) CCR2LRRK2BDKRB1GRIN2BOPRM1
SCHEMBL8617556 0.75 LRRK2 (0.33) LRRK2
SCHEMBL8300408 0.74 KDM4E (0.39)
SCHEMBL8298652 0.69 ITGB3 (0.45) GRIN2B
SCHEMBL8305139 0.68 CDK9 (0.36) LRRK2
SCHEMBL8306016 0.67 GRIN2B (0.38) CCR2RAB9AGRIN2BCHRM4
SCHEMBL8614674 0.66 NAMPT (0.35) RAB9AGRIN2BGPR119

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 2 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed
US-5786371-A INHIBIT AGGREGATION OF BLOOD PLATELETS BOEHRINGER MANNHEIM GMBH (DE) 1998-07-28 US disclosed