SCHEMBL8305658

SCHEMBL8305658

O=C(O)CC1CCC(N2CCC(CCNc3ccnnc3)CC2)CC1

nearest known ligand 0.38

Predicted protein targets (top 16)

geneUniProtsupporting neighboursconfidence
CCNT1 O60563 2/20 0.38
CDK9 P50750 2/20 0.38
HTR2A P28223 1/20 0.37
HRH1 P35367 1/20 0.37
HTR2B P41595 1/20 0.37
ITGB3 P05106 3/20 0.36
ITGA2B P08514 3/20 0.36
FFAR4 Q5NUL3 2/20 0.35
GRIN2B Q13224 1/20 0.34
CXCR3 P49682 1/20 0.34
LRRK2 Q5S007 1/20 0.33
JAK1 P23458 1/20 0.33
TYK2 P29597 1/20 0.33
DGAT1 O75907 1/20 0.33
NAMPT P43490 1/20 0.33
CHRM4 P08173 1/20 0.33

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
SCHEMBL8298652 0.88 ITGB3 (0.45) CCNT1CDK9HTR2AHRH1HTR2B
SCHEMBL8305139 0.86 CDK9 (0.36) CCNT1CDK9HTR2AHRH1HTR2B
SCHEMBL8304380 0.83 DRD3 (0.36) CCNT1CDK9HTR2A
SCHEMBL8301158 0.83 CCR2 (0.35) HTR2AHRH1HTR2BGRIN2BCXCR3
SCHEMBL8300207 0.81 CCR2 (0.34) GRIN2BCXCR3LRRK2CHRM4
SCHEMBL8298648 0.81 CDK9 (0.36) CCNT1CDK9HTR2AHRH1HTR2B
SCHEMBL8300686 0.80 NAMPT (0.43) CCNT1CDK9HTR2AHRH1HTR2B
SCHEMBL8792322 0.77 BDKRB1 (0.31) GRIN2B
SCHEMBL8304874 0.74 FFAR4 (0.41) CCNT1CDK9FFAR4
SCHEMBL8300030 0.73 KDM4E (0.45) CCNT1CDK9HTR2AHRH1HTR2B

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0808306-B1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS ROCHE DIAGNOSTICS GMBH (DE) 1999-08-04 EP disclosed
EP-0808306-A1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS Roche Diagnostics GmbH (DE) 1997-11-26 EP disclosed
WO-1996024586-A1 NEW DERIVATIVES OF PYRIDINE OR PYRIDAZINE, PROCESS FOR PRODUCTION THEREOF AND MEDICAMENTS CONTAINING THESE COMPOUNDS BOEHRINGER MANNHEIM GMBH (DE) 1996-08-15 WO disclosed