SCHEMBL8302463

SCHEMBL8302463

O=C(O)C1(c2cccnc2)CCNCC1

nearest known ligand 0.46

Predicted protein targets (top 18)

geneUniProtsupporting neighboursconfidence
ITGA4 P13612 1/20 0.46
ITGB7 P26010 1/20 0.46
AKR1C1 Q04828 1/20 0.46
OPRM1 P35372 2/20 0.44
MEN1 O00255 1/20 0.44
KMT2A Q03164 1/20 0.44
ALDH1A1 P00352 3/20 0.44
LMNA P02545 1/20 0.44
VNN1 O95497 1/20 0.41
HCAR2 Q8TDS4 2/20 0.40
APP P05067 1/20 0.40
GAA P10253 1/20 0.40
HCAR3 P49019 1/20 0.40
HDAC1 Q13547 1/20 0.39
MKNK1 Q9BUB5 1/20 0.39
MKNK2 Q9HBH9 1/20 0.39
PLOD2 O00469 1/20 0.38
HSD11B1 P28845 1/20 0.38

Click a target to see other patent compounds predicted against it — the reverse direction, in place.

Similar compounds — the chemically nearest patent molecules

Nearest neighbours by Morgan-fingerprint cosine across the patent-compound collection, with each neighbour's top predicted target and the predicted targets it shares with this molecule.

Compoundsimilaritytop predictedshared targets
Hydrochloric Acid SCHEMBL8350428 0.98 ITGA4 (0.45) ITGA4ITGB7AKR1C1OPRM1MEN1
SCHEMBL4825571 0.89 AKR1C1 (0.53) AKR1C1MEN1KMT2AALDH1A1LMNA
Hydrochloric Acid SCHEMBL23778493 0.87 AKR1C1 (0.52) AKR1C1MEN1KMT2AALDH1A1LMNA
SCHEMBL7467936 0.86 OPRM1 (0.45) ITGA4ITGB7OPRM1MEN1KMT2A
SCHEMBL9338162 0.85 AKR1C1 (0.65) ITGA4ITGB7AKR1C1MEN1KMT2A
Hydrochloric Acid SCHEMBL8347400 0.85 OPRM1 (0.44) ITGA4ITGB7OPRM1MEN1KMT2A
SCHEMBL17896072 0.84 AKR1C1 (0.62) ITGA4ITGB7AKR1C1MEN1KMT2A
SCHEMBL8638671 0.83 KMT2A (0.41) ITGA4ITGB7OPRM1MEN1KMT2A
SCHEMBL373567 0.81 AKR1C1 (0.68) AKR1C1OPRM1KMT2AHDAC1HSD11B1
SCHEMBL7338024 0.80 AKR1C1 (0.47) AKR1C1OPRM1KMT2AALDH1A1LMNA

Similarity is cosine over the 2,048-bit Morgan fingerprint (≈ Tanimoto). Identical fingerprints score 1.00.

Patent provenance — the patents this molecule appears in, and who filed them

Claimed or disclosed in 3 patents. claimed = in the patent's claims; disclosed = body only.

PatentTitleAssigneePublishedPriorityFilingCountryStatus
EP-0946548-A1 NOVEL HETEROCYCLIC SUBSTITUTED PYRROLIDINE AMIDE DERIVATIVES HOECHST MARION ROUSSEL, INC. (US) 1999-10-06 EP disclosed
US-5824690-A TREATING ASTHMA, COUGH HOECHST MARION ROUSSEL INC. (US) 1998-10-20 US disclosed
WO-1998027086-A1 NOVEL HETEROCYCLIC SUBSTITUTED PYRROLIDINE AMIDE DERIVATIVES HOECHST MARION ROUSSEL, INC. (US) 1998-06-25 WO disclosed